SCHEMBL28215719

SCHEMBL28215719

CN(C)C1CCN(CCS(=O)(=O)NP(c2ccccc2)c2ccccc2)C1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 5/20 0.47
CCR5 P51681 8/20 0.38
SMYD3 Q9H7B4 1/20 0.37
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37
HDAC1 Q13547 1/20 0.37
HRH2 P25021 1/20 0.36
HRH1 P35367 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36
OPRM1 P35372 1/20 0.36
SIGMAR1 Q99720 1/20 0.36
MAOA P21397 2/20 0.36
MAOB P27338 2/20 0.36
LTA4H P09960 1/20 0.35
CHRM4 P08173 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19507148 0.71 KDM1A (0.39) KDM1ASMYD3HRH2HRH1HRH3
SCHEMBL21300418 0.70 SMYD3 (0.39) KDM1ACCR5SMYD3HRH2HRH1
SCHEMBL19507145 0.70 SMYD3 (0.39) KDM1ACCR5SMYD3HRH2HRH1
SCHEMBL13974454 0.70 SMYD3 (0.39) KDM1ACCR5SMYD3HRH2HRH1
SCHEMBL28215833 0.70 HTR6 (0.38) HTR2AHRH1
SCHEMBL1911332 0.67 LTA4H (0.60) KDM1AHTR2AHTR2CHDAC1OPRM1
SCHEMBL13634431 0.67 LTA4H (0.60) KDM1AHTR2AHTR2CHDAC1OPRM1
SCHEMBL13024536 0.67 LTA4H (0.60) KDM1AHTR2AHTR2CHDAC1OPRM1
SCHEMBL12838076 0.67 KDM1A (0.54) KDM1AHTR2AHRH1OPRM1SIGMAR1
SCHEMBL28215742 0.65 MEN1 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107922362-A 1,3, 4-oxadiazole sulfonamide derivative compounds as histone deacetylase 6 inhibitors and pharmaceutical compositions containing the same 株式会社钟根堂 2018-04-17 CN disclosed