SCHEMBL28217068

SCHEMBL28217068

NCc1cc2cccoc-2c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 6/20 0.58
PRMT6 Q96LA8 1/20 0.49
KEAP1 Q14145 1/20 0.40
NOS3 P29474 2/20 0.39
NOS1 P29475 2/20 0.39
NOS2 P35228 2/20 0.39
CYP2E1 P05181 2/20 0.37
CYP3A4 P08684 2/20 0.37
CYP2D6 P10635 2/20 0.37
CYP2A6 P11509 2/20 0.37
CYP2C9 P11712 2/20 0.37
CYP2B6 P20813 2/20 0.37
CYP2C19 P33261 2/20 0.37
SMARCA2 P51531 1/20 0.37
PBRM1 Q86U86 1/20 0.37
HTR2C P28335 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C8 P10632 1/20 0.35
PSMB5 P28074 1/20 0.34
LOXL2 Q9Y4K0 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL109478 0.85 TAAR1 (0.70) TAAR1PRMT6KEAP1NOS3NOS1
Hydrochloric Acid SCHEMBL1014846 0.83 TAAR1 (0.68) TAAR1PRMT6KEAP1NOS3NOS1
SCHEMBL27569385 0.80 PRMT6 (0.49) TAAR1PRMT6KEAP1SMARCA2PBRM1
SCHEMBL27375459 0.77 TAAR1 (0.59) TAAR1PRMT6HTR2CPOLBALDH1A1
SCHEMBL31456962 0.77 TAAR1 (0.59) TAAR1PRMT6HTR2CPOLBALDH1A1
SCHEMBL112138 0.73 TAAR1 (1.00) TAAR1PRMT6KEAP1CYP2A6HTR2C
SCHEMBL4846415 0.72 TAAR1 (0.54) TAAR1PRMT6KEAP1SMARCA2PBRM1
SCHEMBL10177755 0.72 TAAR1 (0.48) TAAR1CYP2E1CYP3A4CYP2D6CYP2A6
SCHEMBL27559481 0.72 PRMT6 (0.42) TAAR1PRMT6KEAP1CYP3A4CYP2C9
SCHEMBL9454526 0.69 PRMT6 (0.63) TAAR1PRMT6KEAP1PSMB5POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108440515-A Substituted benzofuranyl and benzoxazole based compound and application thereof 卡尔约药物治疗公司 2018-08-24 CN disclosed
CN-105492437-B Substituted benzofuranyl and benzoxazolyl compounds and uses thereof 卡尔约药物治疗公司 2018-05-11 CN disclosed