SCHEMBL28217232

SCHEMBL28217232

CC(C)c1cccc([C@H](C)C2CC2)c1N1CCCC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
TDP1 Q9NUW8 1/20 0.36
GABRA1 P14867 2/20 0.34
GABRG2 P18507 2/20 0.34
GABRB3 P28472 2/20 0.34
FAAH O00519 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
LMNA P02545 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
HPGD P15428 1/20 0.34
TSHR P16473 1/20 0.34
GABRB1 P18505 1/20 0.34
PTGS1 P23219 1/20 0.34
SLC6A2 P23975 1/20 0.34
HTR2C P28335 1/20 0.34
GABRA5 P31644 1/20 0.34
GABRA3 P34903 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28217235 1.00 MEN1 (0.36) MEN1KMT2ATDP1GABRA1GABRG2
SCHEMBL28217215 0.97 KCNQ2 (0.32) MEN1KMT2ATDP1HTR2CHTR2B
SCHEMBL28217217 0.97 KCNQ2 (0.32) MEN1KMT2ATDP1HTR2CHTR2B
SCHEMBL8990154 0.88 GABRA1 (0.43) MEN1KMT2ATDP1GABRA1GABRG2
SCHEMBL28152053 0.86 ALDH1A1 (0.43) MEN1KMT2ATDP1TSHRSLC6A2
SCHEMBL28217231 0.86 CNR2 (0.36) MEN1KMT2ATDP1LMNACYP1A2
SCHEMBL28217234 0.86 CNR2 (0.36) MEN1KMT2ATDP1LMNACYP1A2
SCHEMBL28217676 0.82 LMNA (0.38) MEN1KMT2ATDP1LMNACYP1A2
SCHEMBL28217678 0.82 LMNA (0.38) MEN1KMT2ATDP1LMNACYP1A2
SCHEMBL28217243 0.80 CNR2 (0.33) GABRA1GABRG2GABRB3FAAHCA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108017559-B Benzene ring derivative and application thereof in medicine 四川海思科制药有限公司 2020-08-04 CN disclosed
CN-108017559-A Phenyl ring derivative and its application in medicine 四川海思科制药有限公司 2018-05-11 CN disclosed