SCHEMBL28217704

SCHEMBL28217704

OC1CC(c2ccccc2Br)C1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 3/20 0.48
HTR2C P28335 6/20 0.44
HTR2B P41595 6/20 0.44
BRD4 O60885 1/20 0.43
HTR2A P28223 4/20 0.43
SLC6A2 P23975 2/20 0.43
SLC6A4 P31645 2/20 0.43
SLC6A3 Q01959 1/20 0.43
MAP1LC3B Q9GZQ8 1/20 0.40
HRH3 Q9Y5N1 2/20 0.37
RCOR1 Q9UKL0 1/20 0.36
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
HDAC4 P56524 1/20 0.35
MEN1 O00255 1/20 0.34
GAA P10253 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Formic Acid SCHEMBL28217657 0.91 MAP1LC3B (0.42) KDM1AHTR2CHTR2BBRD4HTR2A
SCHEMBL26834590 0.80 KDM1A (0.41) KDM1AHTR2CHTR2BHTR2ASLC6A2
SCHEMBL22052752 0.80 KDM1A (0.41) KDM1AHTR2CHTR2BHTR2ASLC6A2
SCHEMBL17892133 0.78 KDM1A (0.59) KDM1AHTR2CHTR2BBRD4HTR2A
SCHEMBL31389967 0.77 CHRNB4 (0.43) HTR2CCHRNB4CHRNA3
SCHEMBL10046437 0.77 KDM1A (0.50) KDM1AHTR2CHTR2BBRD4HTR2A
SCHEMBL29427088 0.77 KDM1A (0.50) KDM1AHTR2CHTR2BBRD4HTR2A
SCHEMBL19781088 0.75 TP53 (0.47) KDM1AHTR2CHTR2BBRD4HTR2A
SCHEMBL31389850 0.74 KDM1A (0.50) KDM1AHTR2CHTR2BRCOR1CHRNB4
SCHEMBL18573855 0.74 TP53 (0.50) HTR2CHTR2BHTR2AHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108017643-A A kind of efficient IDO/TDO double inhibitors containing azacyclo- helical structure 中国科学院上海有机化学研究所 2018-05-11 CN disclosed