Formic Acid

Formic Acid

SCHEMBL28217657

O=CO.OC1CC(c2ccccc2Br)C1

nearest known ligand 0.42

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP1LC3B Q9GZQ8 2/20 0.42
KDM1A O60341 2/20 0.42
BRD4 O60885 1/20 0.41
HTR2C P28335 6/20 0.39
HTR2B P41595 6/20 0.39
HTR2A P28223 4/20 0.38
SLC6A2 P23975 2/20 0.38
SLC6A4 P31645 2/20 0.38
SLC6A3 Q01959 1/20 0.38
HDAC4 P56524 1/20 0.34
NPC1 O15118 1/20 0.33
HRH3 Q9Y5N1 2/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
MAPK1 P28482 1/20 0.33
HTT P42858 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28217704 0.91 KDM1A (0.48) MAP1LC3BKDM1ABRD4HTR2CHTR2B
Formic Acid SCHEMBL27536018 0.80 MAP1LC3B (0.43) MAP1LC3BKDM1ABRD4HTR2CHTR2B
SCHEMBL28217656 0.74 MAP1LC3B (0.41) MAP1LC3BKDM1ABRD4HTR2CHTR2B
SCHEMBL26834590 0.73 KDM1A (0.41) KDM1AHTR2CHTR2BHTR2ASLC6A2
SCHEMBL22052752 0.73 KDM1A (0.41) KDM1AHTR2CHTR2BHTR2ASLC6A2
SCHEMBL17892133 0.71 KDM1A (0.59) MAP1LC3BKDM1ABRD4HTR2CHTR2B
Formic Acid SCHEMBL27583413 0.71 HSD11B1 (0.44) NPC1ALDH1A1LMNAMAPK1HTT
SCHEMBL30118017 0.70 MAP1LC3B (0.41) MAP1LC3BKDM1ABRD4HTR2CHTR2B
SCHEMBL31389967 0.70 CHRNB4 (0.43) HTR2C
SCHEMBL10046437 0.69 KDM1A (0.50) MAP1LC3BKDM1ABRD4HTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109890826-A A kind of efficient IDO/TDO double inhibitors containing azacyclo- helical structure 中国科学院上海有机化学研究所 2019-06-14 CN disclosed
CN-108017643-A A kind of efficient IDO/TDO double inhibitors containing azacyclo- helical structure 中国科学院上海有机化学研究所 2018-05-11 CN disclosed