SCHEMBL28218019

SCHEMBL28218019

O=c1ccc2c(-c3ccccc3)ccoc-2c1O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 2/20 0.50
HDAC2 Q92769 2/20 0.50
HDAC8 Q9BY41 2/20 0.50
HDAC6 Q9UBN7 1/20 0.50
PTPRC P08575 1/20 0.44
KDM4E B2RXH2 4/20 0.39
ALDH1A1 P00352 3/20 0.39
MEN1 O00255 2/20 0.39
CYP3A4 P08684 2/20 0.39
KMT2A Q03164 2/20 0.39
HPGD P15428 2/20 0.39
HSD17B10 Q99714 2/20 0.39
MMP1 P03956 1/20 0.39
MMP3 P08254 1/20 0.39
MMP7 P09237 1/20 0.39
MMP9 P14780 1/20 0.39
MMP8 P22894 1/20 0.39
MMP12 P39900 1/20 0.39
MMP13 P45452 1/20 0.39
LMNA P02545 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10900007 0.80 KDM4E (0.48) HDAC4HDAC2HDAC8HDAC6PTPRC
SCHEMBL28218475 0.74 KDM4E (0.50) PTPRCKDM4EALDH1A1HPGDHSD17B10
SCHEMBL23925707 0.73 HDAC4 (0.53) HDAC4HDAC2HDAC8HDAC6PTPRC
SCHEMBL25706171 0.71 CHRM2 (0.51) PTPRCALDH1A1HPGDHSD17B10CHRM2
SCHEMBL28218017 0.70 KDM4E (0.38) PTPRCKDM4EALDH1A1HPGDHSD17B10
SCHEMBL28218014 0.70 KDM4E (0.38) PTPRCKDM4EALDH1A1HPGDHSD17B10
SCHEMBL887941 0.69 CHRM2 (0.50) PTPRCKDM4EALDH1A1MEN1CYP3A4
SCHEMBL31412182 0.68 BACE1 (0.48) HDAC4HDAC2HDAC8HDAC6KDM4E
SCHEMBL21471576 0.68 HDAC4 (1.00) HDAC4HDAC2HDAC8HDAC6ALDH1A1
SCHEMBL12270202 0.66 CHRM2 (0.47) PTPRCKDM4EALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105524034-B Preparation, pharmacological action and the application for treating cerebral ischemia of coumarin derivative 北京大学 2018-08-17 CN disclosed
CN-105566269-B Preparation, pharmacological action and the application for treating itch of coumarin derivative 北京大学 2018-07-10 CN disclosed