SCHEMBL28218017

SCHEMBL28218017

O=c1ccc2c(C(F)(F)F)ccoc-2c1O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.38
LMNA P02545 1/20 0.38
HSPA1A P0DMV8 2/20 0.33
HSPA8 P11142 2/20 0.33
HPGD P15428 2/20 0.33
ALOX15 P16050 2/20 0.33
BRCA1 P38398 2/20 0.33
HSD17B10 Q99714 2/20 0.33
GAPDH P04406 1/20 0.33
GNG2 P59768 1/20 0.33
GNB1 P62873 1/20 0.33
RAPGEF4 Q8WZA2 1/20 0.33
CYP2C9 P11712 1/20 0.33
MAPK1 P28482 1/20 0.33
CYP2C19 P33261 1/20 0.33
HSD17B3 P37058 1/20 0.30
ALDH1A1 P00352 1/20 0.30
CDC25A P30304 1/20 0.30
CDC25B P30305 1/20 0.30
STAT6 P42226 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28218475 0.74 KDM4E (0.50) KDM4ELMNAHSPA1AHSPA8HPGD
SCHEMBL28218014 0.70 KDM4E (0.38) KDM4ELMNAHSPA1AHSPA8HPGD
SCHEMBL28218019 0.70 HDAC4 (0.50) KDM4ELMNAHPGDALOX15HSD17B10
SCHEMBL9625067 0.67 KDM4E (0.50) KDM4ELMNAHPGDMAPK1ALDH1A1
SCHEMBL28218015 0.66 ELANE (0.40) KDM4ELMNAHSPA1AHSPA8HPGD
SCHEMBL23567431 0.62 HSD11B1 (0.46) ALOX15HSD17B10MAPK1CYP2C19ALDH1A1
SCHEMBL16401280 0.62 NOTUM (0.44) HPGDALOX15HSD17B10MAPK1CYP2C19
SCHEMBL10900007 0.62 KDM4E (0.48) KDM4ELMNAHPGDALOX15HSD17B10
SCHEMBL10943763 0.59
SCHEMBL18094477 0.58 CFTR (0.35) KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105524034-B Preparation, pharmacological action and the application for treating cerebral ischemia of coumarin derivative 北京大学 2018-08-17 CN disclosed
CN-105566269-B Preparation, pharmacological action and the application for treating itch of coumarin derivative 北京大学 2018-07-10 CN disclosed
CN-105524034-A Preparation method of coumarin derivative, pharmacological effect of coumarin derivative and use of coumarin derivative in treatment on cerebral ischemia UNIV BEIJING 2016-04-27 CN disclosed