SCHEMBL28218014

SCHEMBL28218014

O=c1ccc2c(CCl)ccoc-2c1O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.38
LMNA P02545 1/20 0.38
AURKA O14965 1/20 0.33
AURKB Q96GD4 1/20 0.33
HSPA1A P0DMV8 2/20 0.33
HSPA8 P11142 2/20 0.33
HPGD P15428 2/20 0.33
ALOX15 P16050 2/20 0.33
BRCA1 P38398 2/20 0.33
HSD17B10 Q99714 2/20 0.33
ALDH1A1 P00352 1/20 0.33
CDC25A P30304 1/20 0.33
CDC25B P30305 1/20 0.33
STAT6 P42226 1/20 0.33
HIF1A Q16665 1/20 0.33
MCL1 Q07820 1/20 0.33
FTO Q9C0B1 1/20 0.31
GAPDH P04406 1/20 0.30
GNG2 P59768 1/20 0.30
GNB1 P62873 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28218015 0.78 ELANE (0.40) KDM4ELMNAHSPA1AHSPA8HPGD
SCHEMBL28218475 0.74 KDM4E (0.50) KDM4ELMNAHSPA1AHSPA8HPGD
SCHEMBL28218019 0.70 HDAC4 (0.50) KDM4ELMNAHPGDALOX15HSD17B10
SCHEMBL28218017 0.70 KDM4E (0.38) KDM4ELMNAHSPA1AHSPA8HPGD
SCHEMBL10900007 0.62 KDM4E (0.48) KDM4ELMNAHPGDALOX15HSD17B10
SCHEMBL11302517 0.60 AURKA (0.54) KDM4EAURKAAURKBHPGDALOX15
SCHEMBL6848551 0.60 KMT2A (0.54) KDM4EHSD17B10ALDH1A1HIF1AMCL1
SCHEMBL10943763 0.59
SCHEMBL11297243 0.58 ELANE (0.51) KDM4ELMNAAURKAAURKBHPGD
SCHEMBL18632773 0.58 ALDH1A1 (0.40) KDM4EHSD17B10ALDH1A1HIF1AMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105524034-B Preparation, pharmacological action and the application for treating cerebral ischemia of coumarin derivative 北京大学 2018-08-17 CN disclosed
CN-105566269-B Preparation, pharmacological action and the application for treating itch of coumarin derivative 北京大学 2018-07-10 CN disclosed