SCHEMBL28220174

SCHEMBL28220174

CCOc1cc(Cl)ccc1C(F)(F)F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.44
HPGD P15428 2/20 0.44
HTT P42858 1/20 0.42
SLC6A4 P31645 4/20 0.42
HTR2A P28223 3/20 0.42
KCNH2 Q12809 1/20 0.42
RXRA P19793 1/20 0.40
RXRB P28702 1/20 0.40
RXRG P48443 1/20 0.40
DRD2 P14416 1/20 0.40
AR P10275 1/20 0.40
MAPT P10636 2/20 0.40
HTR2C P28335 2/20 0.39
HTR2B P41595 2/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.39
MRGPRX4 Q96LA9 2/20 0.39
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
SLC6A2 P23975 1/20 0.38
L3MBTL1 Q9Y468 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18748269 0.84 TSHR (0.45) TSHRHPGDHTTSLC6A4HTR2A
SCHEMBL30628261 0.81 TSHR (0.41) TSHRHPGDHTTRXRARXRB
SCHEMBL17420682 0.81 TSHR (0.41) TSHRHPGDHTTRXRARXRB
SCHEMBL17707963 0.80 AR (0.53) HPGDHTTHTR2ARXRARXRB
SCHEMBL20224866 0.79 DRD2 (0.41) HTTSLC6A4HTR2AKCNH2DRD2
SCHEMBL17420581 0.79 TSHR (0.43) TSHRHPGDHTTHTR2ARXRA
SCHEMBL30628252 0.79 TSHR (0.43) TSHRHPGDHTTHTR2ARXRA
SCHEMBL18833356 0.79 AR (0.43) HPGDHTR2ARXRARXRBRXRG
SCHEMBL28453498 0.79 RXRA (0.40) HPGDHTR2ARXRARXRBRXRG
SCHEMBL2525158 0.77 TSHR (0.56) TSHRHPGDSLC6A4HTR2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104650049-B Substituted pyridine compounds and its application method and purposes 广东东阳光药业有限公司 2018-06-08 CN disclosed