SCHEMBL28229136

SCHEMBL28229136

Nc1cc(Nc2ccccc2-c2ncccn2)c[nH]1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAS2R14 Q9NYV8 3/20 0.38
ADRA1D P25100 1/20 0.38
ADRA1A P35348 1/20 0.38
ADRA1B P35368 1/20 0.38
PIK3CD O00329 1/20 0.35
PIK3CA P42336 1/20 0.35
PIK3CB P42338 1/20 0.35
PIK3CG P48736 1/20 0.35
MAPK14 Q16539 6/20 0.34
KCNK18 Q7Z418 1/20 0.34
AKT1 P31749 1/20 0.33
PIM1 P11309 1/20 0.32
PIM3 Q86V86 1/20 0.32
PIM2 Q9P1W9 1/20 0.32
GRM4 Q14833 1/20 0.32
MAPK10 P53779 2/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
GFER P55789 1/20 0.32
KDM4E B2RXH2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2422607 0.76 MEN1 (0.47) TAS2R14ADRA1DADRA1AADRA1BKCNK18
SCHEMBL23978923 0.64 ADRA1D (0.45) ADRA1DADRA1AADRA1BMAPK10MEN1
SCHEMBL9693871 0.64 ADRA1D (0.45) ADRA1DADRA1AADRA1BMAPK10MEN1
SCHEMBL10599951 0.62 KDM4E (0.45) ADRA1AMEN1KMT2AKDM4EALDH1A1
SCHEMBL1232419 0.61 ALDH1A1 (0.57) MEN1KMT2AKDM4EALDH1A1GAA
SCHEMBL18856198 0.60 PABPC1 (0.43) ADRA1DADRA1AADRA1BMAPK10MEN1
SCHEMBL12853990 0.60 PTPRC (0.44) ADRA1AMEN1KMT2AKDM4EALDH1A1
SCHEMBL29850028 0.59 KMT2A (0.49) ADRA1DADRA1AADRA1BMAPK10MEN1
SCHEMBL18966077 0.59 KMT2A (0.49) ADRA1DADRA1AADRA1BMAPK10MEN1
SCHEMBL22618034 0.59 RET (0.49) MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108191774-A Heterocycle compound, preparation method and use 中国药科大学 2018-06-22 CN claimed
CN-108191774-A Heterocycle compound, preparation method and use 中国药科大学 2018-06-22 CN disclosed