SCHEMBL28229643

SCHEMBL28229643

O=C(O)CC(=O)CCCc1cc(F)cc(F)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP12 P39900 1/20 0.41
HDAC3 O15379 2/20 0.40
HDAC1 Q13547 2/20 0.40
HDAC2 Q92769 2/20 0.40
HDAC8 Q9BY41 2/20 0.40
HDAC6 Q9UBN7 2/20 0.40
HDAC5 Q9UQL6 2/20 0.40
MAPK1 P28482 1/20 0.40
ADRA1A P35348 1/20 0.40
HDAC4 P56524 1/20 0.40
SLC6A3 Q01959 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HDAC7 Q8WUI4 1/20 0.40
HDAC10 Q969S8 1/20 0.40
HDAC11 Q96DB2 1/20 0.40
HDAC9 Q9UKV0 1/20 0.40
LMNA P02545 1/20 0.39
ACLY P53396 1/20 0.37
CYP1A2 P05177 1/20 0.37
FFAR1 O14842 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL316406 0.85 SMN1; SMN2 (0.55) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL28229641 0.83 FFAR1 (0.51) MMP12HDAC3HDAC1HDAC2HDAC8
SCHEMBL27802263 0.82 LMNA (0.56) MMP12HDAC3HDAC1HDAC2HDAC8
SCHEMBL29197998 0.79 MAPT (0.55) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL5907106 0.77 MEN1 (0.41) MMP12FFAR1MEN1KMT2A
SCHEMBL1448093 0.77 KEAP1 (0.52) ACLYFFAR1
SCHEMBL7239123 0.76 HDAC1 (0.70) MMP12HDAC3HDAC1HDAC2HDAC8
SCHEMBL28229640 0.75 FFAR1 (0.42) MMP12HDAC1HDAC7FFAR1
SCHEMBL34471011 0.74 HDAC3 (0.47) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL27816726 0.74 HDAC1 (0.47) MMP12HDAC1HDAC8FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110036014-A A kind of compound and its preparation and application with AXL inhibitory activity 中国科学院上海药物研究所 2019-07-19 CN disclosed
CN-108250200-A A kind of compound and its preparation and application with Axl inhibitory activity 中国科学院上海药物研究所 2018-07-06 CN disclosed