SCHEMBL28239805

SCHEMBL28239805

O=C(OC1CCNCC1)c1ccccc1F

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 7/20 0.50
SLC6A2 P23975 7/20 0.50
SLC6A3 Q01959 3/20 0.50
LMNA P02545 1/20 0.44
KMT2A Q03164 1/20 0.44
CHRM3 P20309 1/20 0.44
CES2 O00748 1/20 0.43
CES1 P23141 1/20 0.43
SLC6A4 P31645 3/20 0.42
SCN1A P35498 2/20 0.42
SCN2A Q99250 2/20 0.42
SCN3A Q9NY46 2/20 0.42
HRH1 P35367 1/20 0.41
ALDH1A1 P00352 2/20 0.41
PTPRF P10586 1/20 0.41
PTPN2 P17706 1/20 0.41
PTPN1 P18031 1/20 0.41
KDM4E B2RXH2 1/20 0.41
POLB P06746 1/20 0.41
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7993233 0.89 CES2 (0.50) LMNAKMT2ACES2CES1SCN1A
SCHEMBL27500253 0.85 KMT2A (0.50) LMNAKMT2ACES2CES1SCN1A
SCHEMBL28239732 0.83 RXFP1 (0.50) HTR1ASLC6A2SLC6A3CHRM3CES2
SCHEMBL7408465 0.81 KMT2A (0.47) LMNAKMT2ACES2CES1SCN1A
SCHEMBL28315283 0.81 SCN1A (0.45) SLC6A2SLC6A3KMT2ACHRM3SLC6A4
SCHEMBL28240607 0.80 MEN1 (0.59) KMT2ACHRM3SCN1ASCN2ASCN3A
SCHEMBL28011429 0.79 SCN1A (0.52) SLC6A2SLC6A3KMT2ACHRM3SLC6A4
SCHEMBL1912949 0.77 CHRNA7 (0.61) KMT2ACHRM3SCN1ASCN2ASCN3A
SCHEMBL29003856 0.77 SLC6A2 (0.53) SLC6A2SLC6A3KMT2ASLC6A4SCN1A
Methylene Chloride SCHEMBL29003874 0.76 MEN1 (0.54) KMT2ACHRM3SCN1ASCN2ASCN3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108456204-B Benzothiazine derivative, and preparation method and application thereof 四川大学 2023-05-26 CN disclosed
CN-108456204-A Benzothiazine derivative and its preparation method and application 四川大学 2018-08-28 CN disclosed