SCHEMBL28242000

SCHEMBL28242000

O=C(CCc1occ2ccccc12)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.44
TDP1 Q9NUW8 3/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
LMNA P02545 1/20 0.44
NR4A2 P43354 1/20 0.44
RAB9A P51151 3/20 0.44
NPC1 O15118 2/20 0.44
CASP3 P42574 1/20 0.44
SENP8 Q96LD8 1/20 0.44
SENP7 Q9BQF6 1/20 0.44
SENP6 Q9GZR1 1/20 0.44
CTNNB1 P35222 3/20 0.42
WNT3A P56704 3/20 0.42
HPGD P15428 2/20 0.41
ALDH1A1 P00352 5/20 0.41
GAA P10253 1/20 0.41
CYP2C19 P33261 1/20 0.41
HDAC3 O15379 1/20 0.41
HDAC4 P56524 1/20 0.41
HDAC1 Q13547 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7859850 0.85 KEAP1 (0.46) MAPTTDP1LMNANR4A2HPGD
SCHEMBL7140950 0.81 EGFR (0.41) MAPTLMNANR4A2GAACYP2C19
SCHEMBL31115079 0.81 MAPT (0.49) MAPTTDP1L3MBTL1LMNARAB9A
SCHEMBL23804836 0.79 CYP1A2 (0.51) MAPTNR4A2ALDH1A1CYP2C19HDAC3
SCHEMBL4413665 0.77 CYP1A2 (0.54) MAPTTDP1L3MBTL1LMNAALDH1A1
SCHEMBL1650809 0.75 KDM4E (0.50) TDP1LMNAHPGDALDH1A1GAA
SCHEMBL2961433 0.74 TDP1 (0.37) MAPTTDP1LMNARAB9AHPGD
SCHEMBL27480509 0.74 S1PR2 (0.41) TDP1HPGDCYP2C19KMT2AKDM4E
SCHEMBL10370767 0.73 KDM4E (0.41) MAPTTDP1L3MBTL1LMNANR4A2
SCHEMBL29580491 0.72 GPR84 (0.68) MAPTTDP1L3MBTL1LMNANR4A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108570027-A A kind of selective PI3K inhibitor for treating tumour 王延娇 2018-09-25 CN disclosed