SCHEMBL28244698

SCHEMBL28244698

CCc1ccc(SC)c(N)c1O

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 1/20 0.43
GABRB2 P47870 1/20 0.43
FEN1 P39748 1/20 0.36
ESR1 P03372 2/20 0.33
ESR2 Q92731 2/20 0.33
NPC1 O15118 1/20 0.30
MAPT P10636 1/20 0.30
RAB9A P51151 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
BACE1 P56817 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9505579 0.79 GABRA1 (0.54) GABRA1GABRB2FEN1ESR1ESR2
SCHEMBL9089334 0.72 GABRA1 (0.41) GABRA1GABRB2NPC1MAPTRAB9A
SCHEMBL21950945 0.72 ALDH1A1 (0.35) NPC1MAPTRAB9ASMN1; SMN2
SCHEMBL45861 0.71 GABRA1 (0.68) GABRA1GABRB2FEN1ESR1ESR2
SCHEMBL8536715 0.68 NPC1 (0.33) NPC1MAPTRAB9A
SCHEMBL9246909 0.68 GAA (0.31) MAPT
SCHEMBL5878543 0.68 HSD17B3 (0.40) GABRA1GABRB2ESR1ESR2MAPT
SCHEMBL5878760 0.68 TYR (0.41) GABRA1GABRB2ESR1ESR2MAPT
SCHEMBL12797849 0.66 POLB (0.41) GABRA1GABRB2MAPTBACE1
Methylamine SCHEMBL27907243 0.66 GABRA1 (0.54) GABRA1GABRB2FEN1ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108658908-B 1,3- bis- replaces ketene compounds and its application 广州必贝特医药技术有限公司 2019-05-10 CN disclosed
CN-108658908-A 1,3- bis- substitution ketene compounds and its application 广州必贝特医药技术有限公司 2018-10-16 CN disclosed