SCHEMBL28246191

SCHEMBL28246191

C#CCc1ccnc(-n2cc(-c3ccncc3)cn2)n1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MELK Q14680 3/20 0.40
KDR P35968 6/20 0.36
FLT1 P17948 2/20 0.36
FLT4 P35916 2/20 0.36
PDE10A Q9Y233 3/20 0.36
ADORA3 P0DMS8 1/20 0.36
ADORA1 P30542 1/20 0.36
DYRK1A Q13627 1/20 0.32
MKNK1 Q9BUB5 2/20 0.32
MKNK2 Q9HBH9 1/20 0.32
CYP3A4 P08684 2/20 0.32
CYP2C9 P11712 2/20 0.32
ALKBH1 Q13686 1/20 0.31
BMP4 P12644 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28042544 0.77 PDE10A (0.45) MELKKDRFLT1FLT4PDE10A
SCHEMBL15905011 0.66 PDE10A (0.74) PDE10A
SCHEMBL28246190 0.62 MELK (0.56) MELKKDRFLT1FLT4DYRK1A
SCHEMBL15293875 0.61 CYP2A6 (0.44) ADORA3ADORA1DYRK1ACYP3A4CYP2C9
SCHEMBL15904208 0.60 PDE10A (0.50) MELKPDE10AADORA3ADORA1CYP3A4
SCHEMBL7106119 0.60 MAPT (0.48) CYP3A4
SCHEMBL12410565 0.59 MELK (0.54) MELKADORA1DYRK1AMKNK1MKNK2
SCHEMBL24921055 0.59 RXRA (0.40) ALKBH1
SCHEMBL6508391 0.58 MELK (0.56) MELKKDRFLT1FLT4MKNK1
SCHEMBL16991685 0.58 MAOA (0.63)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105008346-B Pyrimidine derivatives as phosphodiesterase 10(PDE-10) inhibitors 帕罗生物制药有限公司 2018-11-13 CN disclosed