SCHEMBL28248487

SCHEMBL28248487

CC1CN(C)CCN1Cc1ccc(Br)cc1

nearest known ligand 0.44

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.44
ALDH1A1 P00352 3/20 0.42
KDM4E B2RXH2 2/20 0.40
HRH2 P25021 1/20 0.40
MCHR1 Q99705 1/20 0.39
HRH3 Q9Y5N1 2/20 0.39
RORC P51449 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28248461 0.86 KCNJ1 (0.49) SIGMAR1HRH3
SCHEMBL30361421 0.84 ALDH1A1 (0.60) SIGMAR1ALDH1A1KDM4EHRH2HRH3
SCHEMBL14930169 0.83 MC4R (0.53) SIGMAR1HRH2
SCHEMBL12499953 0.78 KDM4E (0.40) ALDH1A1KDM4EHRH3RORC
SCHEMBL30361428 0.78 KCNJ1 (0.61) SIGMAR1ALDH1A1KDM4EHRH3
SCHEMBL4610176 0.77 ALDH1A1 (0.64) ALDH1A1KDM4EHRH3
SCHEMBL4610173 0.77 ALDH1A1 (0.64) ALDH1A1KDM4EHRH3
SCHEMBL20203572 0.75 ALDH1A1 (0.45) SIGMAR1ALDH1A1HRH3
SCHEMBL20203571 0.75 ALDH1A1 (0.45) SIGMAR1ALDH1A1HRH3
SCHEMBL13046482 0.75 MAPK1 (0.52) SIGMAR1ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108727380-A A kind of BRD4 inhibitor and its preparation and application 中国科学院上海药物研究所 2018-11-02 CN disclosed