SCHEMBL12499953

SCHEMBL12499953

C[C@@H]1CN(C)C[C@H](C)N1Cc1ccc(Br)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.40
ALDH1A1 P00352 2/20 0.40
HDAC1 Q13547 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
HRH3 Q9Y5N1 3/20 0.37
HRH4 Q9H3N8 1/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
BCHE P06276 1/20 0.35
ACHE P22303 1/20 0.35
BACE1 P56817 1/20 0.35
CYP19A1 P11511 1/20 0.35
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
MAPK1 P28482 1/20 0.35
RORC P51449 1/20 0.34
POLB P06746 1/20 0.34
DRD2 P14416 1/20 0.34
LMNA P02545 1/20 0.33
HTT P42858 1/20 0.33
RECQL P46063 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3165429 0.81 MC4R (0.48) ACHE
SCHEMBL3165425 0.81 MC4R (0.48) ACHE
SCHEMBL1427504 0.80 ALDH1A1 (0.42) KDM4EALDH1A1HRH3L3MBTL1BCHE
SCHEMBL29147689 0.80 ALDH1A1 (0.42) KDM4EALDH1A1HRH3L3MBTL1BCHE
SCHEMBL12499770 0.79 ALDH1A1 (0.40) KDM4EALDH1A1CYP19A1CYP11B1CYP11B2
SCHEMBL28248487 0.78 SIGMAR1 (0.44) KDM4EALDH1A1HRH3RORC
SCHEMBL12500077 0.75 HRH3 (0.47) KDM4EALDH1A1HRH3HRH4BCHE
SCHEMBL20432782 0.70 HDAC1 (0.41) KDM4EALDH1A1HDAC1HDAC6L3MBTL1
SCHEMBL20153149 0.70 RET (0.46) HRH3CYP11B1
SCHEMBL16589590 0.70 SIGMAR1 (0.45) KDM4EALDH1A1HRH3HRH4L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012048411-A1 PLK-4 INHIBITORS AND METHOD OF TREATING CANCER WITH SAME UNIVERSITY HEALTH NETWORK (CA) 2012-04-19 WO disclosed