SCHEMBL28252012

SCHEMBL28252012

C[C](C)CN1CCSC1C(=O)NC(CCO)c1ccc(F)cc1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTGFR P43088 1/20 0.44
RPS6KB1 P23443 2/20 0.37
WDR91 A4D1P6 3/20 0.36
KCNK3 O14649 4/20 0.35
CCR5 P51681 1/20 0.34
JAK2 O60674 1/20 0.33
JAK1 P23458 1/20 0.33
TYK2 P29597 1/20 0.33
JAK3 P52333 1/20 0.33
RORC P51449 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3386255 0.82 PTGFR (0.46) PTGFRRPS6KB1WDR91KCNK3CCR5
SCHEMBL22017296 0.81 PTGFR (0.43) PTGFRRPS6KB1WDR91KCNK3CCR5
SCHEMBL18055685 0.78 PTGFR (0.43) PTGFRRPS6KB1CCR5
SCHEMBL13715039 0.78 PTGFR (0.43) PTGFRRPS6KB1CCR5
SCHEMBL3382048 0.73 PTGFR (0.73) PTGFR
SCHEMBL27049055 0.73 PTGFR (0.73) PTGFR
SCHEMBL3381107 0.73 PTGFR (0.73) PTGFR
SCHEMBL22017295 0.72 PTGFR (0.58) PTGFRRPS6KB1CCR5
SCHEMBL3382831 0.71 PTGFR (0.64) PTGFR
SCHEMBL7045396 0.71 PRKACA (0.40) PTGFRRPS6KB1WDR91CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108779087-A The Valine ester and its salt form, crystal polymorph of hydroxypropyl thiazolidine carboxamide derivative 默克雪兰诺有限公司 2018-11-09 CN disclosed