SCHEMBL28252589

SCHEMBL28252589

N#Cc1nn(Cc2cccnc2)c2cccc(F)c12

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 3/20 0.42
GRIN1 Q05586 6/20 0.41
GRIN2B Q13224 6/20 0.41
ALDH1A1 P00352 2/20 0.40
KDM4E B2RXH2 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
PKM P14618 1/20 0.40
APP P05067 3/20 0.38
SNCA P37840 3/20 0.38
RORC P51449 1/20 0.38
AR P10275 2/20 0.37
SCN9A Q15858 1/20 0.37
CHRNB2 P17787 1/20 0.37
CHRNA4 P43681 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23162012 0.81 P2RX7 (0.42) P2RX7GRIN1GRIN2BALDH1A1KDM4E
SCHEMBL20534347 0.80 APP (0.48) P2RX7ALDH1A1PKMAPPSNCA
SCHEMBL28956925 0.77 GRIN1 (0.43) P2RX7GRIN1GRIN2BALDH1A1KDM4E
SCHEMBL20534644 0.77 GRIN1 (0.43) P2RX7GRIN1GRIN2BALDH1A1PKM
SCHEMBL23161999 0.74 ALDH1A1 (0.39) P2RX7GRIN1GRIN2BALDH1A1KDM4E
SCHEMBL186021 0.69 GRIN1 (0.44) GRIN1GRIN2BALDH1A1RORC
SCHEMBL16252841 0.68 ALDH1A1 (0.43) ALDH1A1KDM4ERORC
SCHEMBL15552018 0.68 CSF1R (0.50) P2RX7ALDH1A1KDM4EPKMCHRNB2
SCHEMBL23161955 0.68 KCNK13 (0.37) GRIN1GRIN2B
SCHEMBL20140391 0.67 BUB1 (0.48) PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108727340-A Fluorine-substituted indazole compounds and application thereof 广东东阳光药业有限公司 2018-11-02 CN disclosed