SCHEMBL28253552

SCHEMBL28253552

CS(=O)(=O)O.Cc1cn(C)c(C)n1

nearest known ligand 0.39

Known targets — ChEMBL curated mechanism

ABL1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB2AGTR1BCL2BCL2A1BCL2L1BCL2L10BCL2L2BCRBRAFCHRM1CHRNA10CHRNA9DRD1DRD2DRD3DRD4DRD5EGFRF2FLT1FLT4GCKGHSRGNRHRGRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BHTR1AHTR1BHTR1DHTR2AHTR2CHTR3AIDH2KDRKITMAOBMCL1MTTPPP4HBPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PIKFYVEROCK1ROCK2SLC18A2SLC6A2SLC6A3SLC6A4TACR1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8gyrAgyrBparCparEpol

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.39
TDP1 Q9NUW8 1/20 0.38
LMNA P02545 1/20 0.38
NLRP3 Q96P20 1/20 0.36
TSHR P16473 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
KDM4E B2RXH2 2/20 0.33
THRB P10828 1/20 0.33
RXFP1 Q9HBX9 1/20 0.32
CCNE1 P24864 1/20 0.31
CDK2 P24941 1/20 0.31
PTGDR2 Q9Y5Y4 1/20 0.31
PTGS2 P35354 1/20 0.30
GAA P10253 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18879399 0.86 TDP1 (0.38) ALDH1A1TDP1LMNANLRP3TSHR
SCHEMBL486467 0.84
Iodide SCHEMBL3791317 0.82
Water SCHEMBL7594635 0.82
Acetic Acid SCHEMBL28272591 0.81 TSHR (0.38) ALDH1A1LMNANLRP3TSHRNPSR1
Formamide SCHEMBL23636189 0.77 ALDH1A1 (0.33) ALDH1A1TSHRNPSR1
SCHEMBL2702033 0.77 TDP1 (0.45) TDP1LMNANLRP3KDM4ETHRB
SCHEMBL27833603 0.75 POLB (0.34) ALDH1A1TSHR
Hydrochloric Acid SCHEMBL27570535 0.75 TDP1 (0.44) TDP1LMNANLRP3KDM4ETHRB
SCHEMBL4946725 0.73

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109504015-A Electrochromic polymeric compounds material based on combined strategy and prepare electrochromic device 常州铱视光电科技有限公司 2019-03-22 CN claimed
CN-109504015-A Electrochromic polymeric compounds material based on combined strategy and prepare electrochromic device 常州铱视光电科技有限公司 2019-03-22 CN disclosed
CN-108795407-A Based on the electroluminescent sour electrochromic material acted on and prepare electrochromic device 常州铱视光电科技有限公司 2018-11-13 CN disclosed