SCHEMBL28258271

SCHEMBL28258271

C=CC(c1ccccc1)c1cccc(C(N)=O)c1C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 9/20 0.36
MAPT P10636 6/20 0.36
CYP3A4 P08684 3/20 0.36
ALOX15 P16050 3/20 0.36
RPS6KB1 P23443 3/20 0.36
AURKA O14965 2/20 0.36
AURKB Q96GD4 1/20 0.36
BCAT2 O15382 1/20 0.36
IRAK4 Q9NWZ3 1/20 0.36
KEAP1 Q14145 1/20 0.36
NFE2L2 Q16236 1/20 0.36
HPGD P15428 6/20 0.35
ALDH1A1 P00352 4/20 0.35
HSD17B10 Q99714 3/20 0.35
LMNA P02545 3/20 0.35
USP2 O75604 2/20 0.35
TP53 P04637 2/20 0.35
TDP1 Q9NUW8 2/20 0.35
ALOX12 P18054 1/20 0.35
MEN1 O00255 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9542306 0.86 KDM4E (0.41) KDM4EMAPTCYP3A4ALOX15BCAT2
SCHEMBL6278245 0.77 ALDH1A1 (0.49) KDM4EMAPTCYP3A4ALOX15HPGD
SCHEMBL28692019 0.75 ALDH1A1 (0.44) KDM4EMAPTCYP3A4ALOX15HPGD
SCHEMBL29129651 0.74 CTSD (0.41) KDM4EMAPTCYP3A4ALOX15HPGD
SCHEMBL5682092 0.73 MAPT (0.39) KDM4EMAPTCYP3A4ALOX15HPGD
SCHEMBL24692389 0.73 IRAK4 (0.44) KDM4EMAPTCYP3A4IRAK4KEAP1
SCHEMBL27432511 0.73 AKR1C3 (0.46) KDM4EMAPTCYP3A4ALOX15HPGD
SCHEMBL19437356 0.72 CXCR2 (0.44) KDM4EHPGDALDH1A1HSD17B10LMNA
SCHEMBL19437462 0.72 LMNA (0.44) KDM4EMAPTCYP3A4ALOX15HPGD
SCHEMBL3792769 0.72 AKR1C3 (0.44) KDM4EMAPTCYP3A4ALOX15ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108884083-A Benzo [ B ] furans as bromodomain inhibitors 葛兰素史克知识产权第二有限公司 2018-11-23 CN disclosed