SCHEMBL2825829

SCHEMBL2825829

Cc1cc(Sc2cc(C#Cc3nccs3)cc(C#Cc3nccs3)c2)ccc1[O]

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 3/20 0.43
ACACB O00763 1/20 0.37
PDE10A Q9Y233 2/20 0.35
KDM4E B2RXH2 1/20 0.33
HAO1 Q9UJM8 2/20 0.32
NPC1 O15118 3/20 0.32
RAB9A P51151 3/20 0.32
CFTR P13569 1/20 0.32
POLB P06746 1/20 0.32
MAPT P10636 1/20 0.32
PPARG P37231 1/20 0.31
NCOR2 Q9Y618 1/20 0.31
FBP1 P09467 1/20 0.31
ALDH1A1 P00352 1/20 0.30
PKM P14618 1/20 0.30
HPGD P15428 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2068873 0.80 PPARD (0.48) PPARG
SCHEMBL2820978 0.77 GRM5 (0.44) GRM5NPC1RAB9APOLB
SCHEMBL2069218 0.76 PPARA (0.40) GRM5ACACBPDE10AHAO1NPC1
SCHEMBL2068786 0.74 PPARD (0.46) PPARG
SCHEMBL2821756 0.71 GRM5 (0.41) GRM5NPC1RAB9AMAPT
SCHEMBL2827409 0.69 GRM5 (0.47) GRM5HAO1
SCHEMBL30278513 0.66 GRM5 (0.68) GRM5ACACBPDE10AKDM4EHAO1
SCHEMBL2822191 0.66 GRM5 (0.43) GRM5MAPTPPARGALDH1A1HPGD
SCHEMBL6311520 0.65 GRM5 (0.65) GRM5ACACBPDE10AHAO1
SCHEMBL15870993 0.64 GRM5 (0.68) GRM5ACACBPDE10AHAO1FBP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1745003-B1 NOVEL COMPOUNDS, THEIR PREPARATION AND USE HIGH POINT PHARMACEUTICALS LLC (US) 2010-10-27 EP claimed