SCHEMBL28260511

SCHEMBL28260511

COC(=O)C1(C(F)F)CCc2ccc(Cl)cc2C1=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.40
F7 P08709 1/20 0.37
PARP1 P09874 1/20 0.37
F3 P13726 1/20 0.37
PARP10 Q53GL7 1/20 0.37
SPR P35270 1/20 0.36
TRPV1 Q8NER1 2/20 0.35
TSHR P16473 1/20 0.34
ALDH1A1 P00352 2/20 0.34
DGAT1 O75907 3/20 0.34
SRD5A1 P18405 3/20 0.33
SRD5A2 P31213 2/20 0.33
CNR2 P34972 1/20 0.33
ADRA1D P25100 1/20 0.33
ADRA1A P35348 1/20 0.33
ADRA1B P35368 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
GAA P10253 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28261809 0.88 TSHR (0.41) SMN1; SMN2PARP1PARP10TSHRSRD5A1
SCHEMBL28351697 0.86 SMN1; SMN2 (0.53) SMN1; SMN2ALDH1A1
SCHEMBL28355728 0.83 HTR2A (0.43) SMN1; SMN2TSHRALDH1A1CYP1A2CYP3A4
SCHEMBL28355808 0.81 SMN1; SMN2 (0.38) SMN1; SMN2ALDH1A1SRD5A1SRD5A2CYP1A2
SCHEMBL28260480 0.81 SMN1; SMN2 (0.43) SMN1; SMN2ALDH1A1CYP3A4GAA
SCHEMBL28260461 0.80 SMN1; SMN2 (0.48) SMN1; SMN2TSHRDGAT1SRD5A1CYP2C19
SCHEMBL28260554 0.79 SMN1; SMN2 (0.47) SMN1; SMN2PARP10TSHRALDH1A1DGAT1
SCHEMBL28351995 0.79 SMN1; SMN2 (0.66) SMN1; SMN2ALDH1A1DGAT1GAA
SCHEMBL28261777 0.76 TSHR (0.42) SMN1; SMN2TSHRALDH1A1CYP3A4GAA
SCHEMBL28352016 0.74 KDM4E (0.40) SMN1; SMN2PARP1PARP10TSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108997183-B Difluoromethylation reagent and preparation method and application thereof 深圳大学 2020-02-07 CN claimed
CN-108997183-A A kind of difluoromethyl reagent and the preparation method and application thereof 深圳大学 2018-12-14 CN disclosed