SCHEMBL28263243

SCHEMBL28263243

C1=C2NCCC2CN1Cc1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.38
ALDH1A1 P00352 3/20 0.36
FUCA1 P04066 2/20 0.36
ACHE P22303 2/20 0.36
TDP1 Q9NUW8 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C19 P33261 1/20 0.36
MAPT P10636 1/20 0.35
POLB P06746 1/20 0.35
CCR3 P51677 1/20 0.35
GSK3A P49840 1/20 0.35
GSK3B P49841 1/20 0.35
HPGD P15428 1/20 0.35
TSHR P16473 1/20 0.35
BCHE P06276 1/20 0.35
BACE1 P56817 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12821980 0.91 ALDH1A1 (0.37) SIGMAR1ALDH1A1FUCA1TDP1CYP1A2
SCHEMBL28145547 0.86 SIGMAR1 (0.42) SIGMAR1ALDH1A1ACHETDP1MAPT
SCHEMBL28145498 0.77 SIGMAR1 (0.44) SIGMAR1ALDH1A1FUCA1ACHETDP1
Hydrochloric Acid SCHEMBL1904419 0.73 LTA4H (0.55)
SCHEMBL3058629 0.70 SMN1; SMN2 (0.46) CYP2D6CYP2C19
SCHEMBL1749081 0.70 GSK3A (0.40) ALDH1A1FUCA1TDP1GSK3AGSK3B
SCHEMBL3021140 0.69 SIGMAR1 (0.38) SIGMAR1FUCA1GSK3AGSK3BHPGD
SCHEMBL5540890 0.68 SIGMAR1 (0.46) SIGMAR1ALDH1A1FUCA1ACHECYP1A2
SCHEMBL7234813 0.65 SIGMAR1 (0.44) SIGMAR1
Hydrochloric Acid SCHEMBL21815558 0.64

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105085525-B Isoquinolin sulfonyl derivative as RHO kinase inhibitor 南京明德新药研发股份有限公司 2019-01-04 CN disclosed