SCHEMBL2826445

SCHEMBL2826445

Cc1nc2c(OC(F)(F)F)cccc2c(-c2cccc(Cl)c2)c1C(=O)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.48
MAPT P10636 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
FABP3 P05413 1/20 0.43
FABP4 P15090 1/20 0.43
NR1H2 P55055 4/20 0.40
NR1H3 Q13133 4/20 0.40
CTSA P10619 2/20 0.39
ALOX15 P16050 1/20 0.39
HTT P42858 3/20 0.38
KDM4E B2RXH2 3/20 0.38
LMNA P02545 1/20 0.38
PLA2G2A P14555 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.38
MAP2 P11137 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
NR1I3 Q14994 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2825663 0.89 KMT2A (0.41) FABP3FABP4NR1H2CTSAHTT
SCHEMBL2821965 0.88 FABP3 (0.39) FABP3FABP4CTSAHTTKDM4E
SCHEMBL2822034 0.82 FABP3 (0.53) GAAMAPTNPSR1FABP3FABP4
SCHEMBL2824267 0.81 ALDH1A1 (0.48) GAAMAPTNPSR1FABP3FABP4
SCHEMBL2825609 0.80 SMN1; SMN2 (0.44) GAAMAPTNPSR1FABP3FABP4
SCHEMBL2824685 0.79 KDM4E (0.41) MAPTNPSR1FABP3FABP4NR1H2
SCHEMBL2824278 0.78 MRGPRX1 (0.38) HTT
SCHEMBL2824252 0.78 FABP3 (0.38) GAAMAPTNPSR1FABP3FABP4
SCHEMBL2824206 0.76 DHODH (0.37) NR1H2NR1H3PTGDR2
SCHEMBL1125943 0.75 GAA (0.64) GAAMAPTNPSR1NR1H2NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1809605-B1 QUINOLINES AS ALLOSTERIC ENHANCERS OF THE GABA-B RECEPTORS HOFFMANN LA ROCHE (CH) 2010-08-11 EP claimed