SCHEMBL2824685

SCHEMBL2824685

CC(=O)c1c(C)nc2c(OC(F)(F)F)cccc2c1-c1ccc(Cl)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.41
ALDH1A1 P00352 4/20 0.41
KMT2A Q03164 4/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
RAB9A P51151 3/20 0.41
MEN1 O00255 2/20 0.41
NPC1 O15118 2/20 0.41
PKM P14618 1/20 0.41
NPSR1 Q6W5P4 3/20 0.39
FABP3 P05413 1/20 0.39
FABP4 P15090 1/20 0.39
NR1H2 P55055 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.38
LMNA P02545 1/20 0.38
MAPT P10636 1/20 0.38
HTT P42858 1/20 0.38
TNKS O95271 1/20 0.38
TNKS2 Q9H2K2 1/20 0.38
PARP2 Q9UGN5 1/20 0.38
HPGD P15428 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2824252 0.90 FABP3 (0.38) KDM4EALDH1A1KMT2ASMN1; SMN2RAB9A
SCHEMBL2824267 0.90 ALDH1A1 (0.48) KDM4EALDH1A1KMT2ASMN1; SMN2RAB9A
SCHEMBL2825663 0.89 KMT2A (0.41) KDM4EALDH1A1KMT2AFABP3FABP4
SCHEMBL2824278 0.89 MRGPRX1 (0.38) ALDH1A1HTTCYP2C9POLB
SCHEMBL2823538 0.83 FABP3 (0.44) KDM4EALDH1A1KMT2ASMN1; SMN2RAB9A
SCHEMBL2823282 0.81 ENPP1 (0.39) KDM4EALDH1A1KMT2ASMN1; SMN2MEN1
SCHEMBL2821965 0.80 FABP3 (0.39) KDM4EKMT2ASMN1; SMN2FABP3FABP4
SCHEMBL2825609 0.80 SMN1; SMN2 (0.44) KDM4EALDH1A1KMT2ASMN1; SMN2RAB9A
SCHEMBL2826082 0.79 ENPP1 (0.43) KDM4EALDH1A1KMT2ASMN1; SMN2MEN1
SCHEMBL2826445 0.79 GAA (0.48) KDM4EKMT2ASMN1; SMN2MEN1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1809605-B1 QUINOLINES AS ALLOSTERIC ENHANCERS OF THE GABA-B RECEPTORS HOFFMANN LA ROCHE (CH) 2010-08-11 EP claimed