SCHEMBL2824252

SCHEMBL2824252

Cc1nc2c(OC(F)(F)F)cccc2c(-c2ccc(Cl)cc2)c1C(=O)C(F)(F)F

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FABP3 P05413 1/20 0.38
FABP4 P15090 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.38
TNKS O95271 1/20 0.37
TNKS2 Q9H2K2 1/20 0.37
PARP2 Q9UGN5 1/20 0.37
NR1H2 P55055 1/20 0.36
DHODH Q02127 1/20 0.36
MAP2 P11137 1/20 0.35
ANO1 Q5XXA6 1/20 0.35
ADORA2A P29274 1/20 0.35
ADORA1 P30542 1/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
GAA P10253 1/20 0.34
MAPT P10636 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
CTSA P10619 2/20 0.34
PLA2G2A P14555 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2823282 0.91 ENPP1 (0.39) PTGDR2TNKSTNKS2PARP2DHODH
SCHEMBL2824685 0.90 KDM4E (0.41) FABP3FABP4PTGDR2TNKSTNKS2
SCHEMBL2825609 0.90 SMN1; SMN2 (0.44) FABP3FABP4NR1H2DHODHADORA2A
SCHEMBL2821965 0.90 FABP3 (0.39) FABP3FABP4PTGDR2MAP2ADORA2A
SCHEMBL2826082 0.88 ENPP1 (0.43) TNKSTNKS2PARP2ADORA2AADORA1
SCHEMBL2824206 0.88 DHODH (0.37) PTGDR2NR1H2DHODHADORA2AADORA1
SCHEMBL2825639 0.87 NR1H2 (0.40) PTGDR2NR1H2
SCHEMBL2826114 0.83 CYP1A2 (0.39) TNKSTNKS2PARP2NR1H2DHODH
SCHEMBL2824267 0.80 ALDH1A1 (0.48) FABP3FABP4NR1H2SMN1; SMN2GAA
SCHEMBL2825663 0.80 KMT2A (0.41) FABP3FABP4PTGDR2NR1H2MAP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1809605-B1 QUINOLINES AS ALLOSTERIC ENHANCERS OF THE GABA-B RECEPTORS HOFFMANN LA ROCHE (CH) 2010-08-11 EP claimed