SCHEMBL28265035

SCHEMBL28265035

O=S(=O)(c1ccc2ccccc2n1)C1CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
NCF1 P14598 2/20 0.38
CYP1A2 P05177 2/20 0.38
NOS2 P35228 1/20 0.38
BACE1 P56817 1/20 0.38
CA12 O43570 1/20 0.38
CA9 Q16790 1/20 0.38
MGAM O43451 1/20 0.38
ALDH1A1 P00352 2/20 0.38
CYP3A4 P08684 2/20 0.38
MEN1 O00255 1/20 0.38
TP53 P04637 1/20 0.38
MAPT P10636 1/20 0.38
MAPK1 P28482 1/20 0.38
KMT2A Q03164 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HIF1A Q16665 1/20 0.38
HRH3 Q9Y5N1 2/20 0.37
HDAC1 Q13547 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Quinoline SCHEMBL28264935 0.91 ALDH1A1 (0.50) NPC1RAB9ACYP1A2ALDH1A1CYP3A4
SCHEMBL3213359 0.89 CYP3A4 (0.42) NPC1RAB9ACYP1A2ALDH1A1CYP3A4
SCHEMBL3219342 0.78 CYP3A4 (0.42) RAB9AALDH1A1CYP3A4MAPK1SMN1; SMN2
SCHEMBL7028380 0.75 HTR2A (0.52)
SCHEMBL329691 0.75 CYP1A2 (0.50) NCF1CYP1A2NOS2BACE1CA12
SCHEMBL11679239 0.75 NCF1 (0.45) NPC1RAB9ANCF1CYP1A2NOS2
SCHEMBL546320 0.73 MGAM (0.47) NPC1RAB9ANCF1CYP1A2NOS2
SCHEMBL14194322 0.73 NCF1 (0.43) NPC1RAB9ANCF1CYP1A2NOS2
SCHEMBL645967 0.73 NCF1 (0.48) NPC1RAB9ANCF1CYP1A2NOS2
SCHEMBL5609339 0.73 NCF1 (0.43) NPC1RAB9ANCF1CYP1A2NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109134364-B Synthesis method of 2-aliphatic sulfonyl quinoline derivative 中南大学 2020-05-05 CN disclosed
CN-109134364-A A kind of synthetic method of 2- aliphaticsulfonyl quinoline 中南大学 2019-01-04 CN disclosed