SCHEMBL28274241

SCHEMBL28274241

C[C@@H]1CN(c2cnccn2)CCN1C(=O)OC(C)(C)C

nearest known ligand 0.60

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 5/20 0.60
GRM1 Q13255 7/20 0.59
MAP4K4 O95819 1/20 0.55
HDAC1 Q13547 1/20 0.52
KDM4E B2RXH2 1/20 0.45
SLC6A9 P48067 1/20 0.42
RXFP1 Q9HBX9 1/20 0.41
TP53 P04637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28274242 1.00 GPR119 (0.60) GPR119GRM1MAP4K4HDAC1KDM4E
SCHEMBL12100832 0.83 GRM1 (0.64) GPR119GRM1MAP4K4HDAC1KDM4E
SCHEMBL12100833 0.83 GRM1 (0.64) GPR119GRM1MAP4K4HDAC1KDM4E
SCHEMBL28966643 0.83 MAP4K4 (0.52) GPR119GRM1MAP4K4HDAC1SLC6A9
SCHEMBL28966679 0.83 MAP4K4 (0.52) GPR119GRM1MAP4K4HDAC1SLC6A9
SCHEMBL28966641 0.83 MAP4K4 (0.52) GPR119GRM1MAP4K4HDAC1SLC6A9
SCHEMBL23560874 0.82 MAP4K4 (0.54) GPR119GRM1MAP4K4HDAC1
SCHEMBL21460229 0.82 MAP4K4 (0.54) GPR119GRM1MAP4K4HDAC1
SCHEMBL31104870 0.82 MAP4K4 (0.59) GPR119GRM1MAP4K4HDAC1
SCHEMBL21484275 0.82 MAP4K4 (0.59) GPR119GRM1MAP4K4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109311867-A Conjugate comprising RIPK2 inhibitor 葛兰素史克知识产权开发有限公司 2019-02-05 CN disclosed