SCHEMBL28274284

SCHEMBL28274284

CC1(c2ccc(I)cc2)NCCc2ccccc21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.39
MEN1 O00255 1/20 0.39
CYP2D6 P10635 1/20 0.39
ALOX15 P16050 1/20 0.39
CYP2C19 P33261 1/20 0.39
KMT2A Q03164 1/20 0.39
GRIN2D O15399 1/20 0.39
GRIN3B O60391 1/20 0.39
BCHE P06276 1/20 0.39
CHRM5 P08912 1/20 0.39
TSHR P16473 1/20 0.39
ALOX12 P18054 1/20 0.39
NFKB1 P19838 1/20 0.39
MAPK1 P28482 1/20 0.39
PRCP P42785 1/20 0.39
GRIN1 Q05586 1/20 0.39
GRIN2A Q12879 1/20 0.39
GRIN2B Q13224 1/20 0.39
GRIN2C Q14957 1/20 0.39
GRIN3A Q8TCU5 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9374419 0.87 CYP3A4 (0.42) CYP3A4MEN1CYP2D6ALOX15CYP2C19
Hydrochloric Acid SCHEMBL6021932 0.85 CYP3A4 (0.41) CYP3A4MEN1CYP2D6ALOX15CYP2C19
Hydrochloric Acid SCHEMBL9376448 0.84 OPRM1 (0.41) CYP3A4MEN1CYP2D6ALOX15CYP2C19
Hydrochloric Acid SCHEMBL9377127 0.83 HTR2A (0.41) CYP3A4MEN1CYP2D6ALOX15CYP2C19
Hydrochloric Acid SCHEMBL9375136 0.83 CYP3A4 (0.38) CYP3A4MEN1CYP2D6ALOX15CYP2C19
Hydrochloric Acid SCHEMBL9374439 0.81 ATM (0.44)
SCHEMBL19565427 0.81 ALDH1A1 (0.36) CYP3A4ALOX12HSD17B10
SCHEMBL19454255 0.80 DRD2 (0.41) CYP3A4ALOX12HSD17B10
Hydrochloric Acid SCHEMBL9375331 0.78 EDNRB (0.44) CYP3A4MEN1CYP2D6ALOX15CYP2C19
SCHEMBL19439341 0.77 KDM1A (0.41) KDM1AHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109219604-A Tetrahydroisoquinoline estrogenic agents and application thereof 豪夫迈·罗氏有限公司 2019-01-15 CN disclosed