SCHEMBL28280694

SCHEMBL28280694

COC(=O)c1c(C2CC2)nc2ccccc2c1N

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.50
BCHE P06276 1/20 0.50
HSD17B10 Q99714 3/20 0.49
KMT2A Q03164 3/20 0.49
MEN1 O00255 2/20 0.49
TP53 P04637 1/20 0.49
KDM4E B2RXH2 3/20 0.48
ALDH1A1 P00352 3/20 0.48
HPGD P15428 3/20 0.48
POLB P06746 1/20 0.48
MAPT P10636 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.47
TSHR P16473 1/20 0.44
MAPK1 P28482 1/20 0.44
GABRP O00591 2/20 0.43
GABRD O14764 2/20 0.43
GABRA1 P14867 2/20 0.43
GABRB1 P18505 2/20 0.43
GABRG2 P18507 2/20 0.43
GABRB3 P28472 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28281977 0.86 KDM4E (0.50) ACHEBCHEHSD17B10KMT2AMEN1
SCHEMBL8574356 0.79 HSD17B10 (0.55) ACHEHSD17B10KMT2AMEN1TP53
SCHEMBL7649523 0.79 HSD17B10 (0.72) HSD17B10KMT2AMEN1TP53KDM4E
SCHEMBL6924495 0.78 ACHE (0.49) ACHEBCHEHSD17B10TP53KDM4E
SCHEMBL356302 0.78 PRKAA2 (0.61) KMT2AMEN1TP53KDM4EALDH1A1
SCHEMBL618360 0.76 ALDH1A1 (0.53) HSD17B10KMT2AMEN1TP53KDM4E
SCHEMBL28281976 0.73 ACHE (0.47) ACHEBCHEHSD17B10KMT2AMEN1
SCHEMBL2443270 0.73 MEN1 (0.71) KMT2AMEN1KDM4EALDH1A1HPGD
SCHEMBL38662586 0.73 MEN1 (0.71) KMT2AMEN1KDM4EALDH1A1HPGD
SCHEMBL14916910 0.72 FABP4 (0.60) KMT2AMEN1KDM4EMAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109422681-A A kind of preparation method of Pitavastatin Calcium intermediate 浙江京新药业股份有限公司 2019-03-05 CN disclosed