SCHEMBL28285545

SCHEMBL28285545

COc1ccc(COC(=O)NC2CC2)cc1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.70
PKM P14618 2/20 0.70
HTT P42858 2/20 0.70
ALDH1A1 P00352 5/20 0.59
GAA P10253 1/20 0.59
EPHX2 P34913 1/20 0.57
TSHR P16473 1/20 0.57
EPHX1 P07099 1/20 0.57
NPC1 O15118 1/20 0.53
RAB9A P51151 1/20 0.53
CA1 P00915 2/20 0.52
CA2 P00918 2/20 0.52
ACHE P22303 2/20 0.52
ATM Q13315 1/20 0.51
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
HPGD P15428 1/20 0.51
CYP2C19 P33261 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22104103 0.93 EPHX2 (0.68) SMN1; SMN2PKMHTTALDH1A1EPHX2
SCHEMBL16018991 0.85 PKM (0.60) SMN1; SMN2PKMHTTALDH1A1EPHX2
SCHEMBL17658614 0.81 ALDH1A1 (0.62) SMN1; SMN2PKMHTTALDH1A1GAA
SCHEMBL3948461 0.81 ALDH1A1 (0.85) ALDH1A1GAATSHREPHX1CA1
SCHEMBL381922 0.81 ALDH1A1 (0.85) ALDH1A1GAATSHREPHX1CA1
SCHEMBL3948456 0.81 ALDH1A1 (0.85) ALDH1A1GAATSHREPHX1CA1
Methoxyamine SCHEMBL5122725 0.81 TSHR (0.75) ALDH1A1GAATSHREPHX1CA1
SCHEMBL15495455 0.80 PKM (0.60) SMN1; SMN2PKMHTTALDH1A1GAA
Hydrochloric Acid SCHEMBL28135182 0.80 ALDH1A1 (0.83) ALDH1A1GAATSHREPHX1CA1
SCHEMBL1675909 0.79 EPHX2 (0.59) SMN1; SMN2PKMHTTALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105153028-B Compound as c-Met kinase inhibitor 南京爱德程医药科技有限公司 2019-03-26 CN disclosed
CN-104936946-A Process for preparing antitumor agent 6- (7- ((1-aminocyclopropyl) methoxy) -6-methoxyquinolin-4-yloxy) -N-methyl-1-naphthamide and crystal thereof ADVENCHEN PHARMACEUTICALS LLC 2015-09-23 CN disclosed