SCHEMBL28286273

SCHEMBL28286273

Nc1cncc(NC=O)c1

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
KDM4E B2RXH2 1/20 0.39
LMNA P02545 1/20 0.39
DDO Q99489 1/20 0.39
KCNH2 Q12809 1/20 0.39
SCN5A Q14524 1/20 0.39
SCN9A Q15858 1/20 0.39
PIK3CB P42338 1/20 0.31
CYP11B1 P15538 1/20 0.30
CYP11B2 P19099 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27918809 0.84 ALDH1A1 (0.44) ALDH1A1MEN1KMT2AKDM4ELMNA
SCHEMBL18925305 0.78 KCNH2 (0.38) ALDH1A1MEN1KMT2AKDM4ELMNA
SCHEMBL3690367 0.75 ALDH1A1 (0.44) ALDH1A1LMNA
Pyridine SCHEMBL28061631 0.73 ALDH1A1 (0.45) ALDH1A1MEN1KMT2AKDM4E
Hydrochloric Acid SCHEMBL7638318 0.72 MEN1 (0.33) ALDH1A1MEN1KMT2APIK3CB
SCHEMBL23940274 0.72 RAF1 (0.37) ALDH1A1MEN1KMT2AKCNH2CYP11B1
SCHEMBL22606743 0.71
SCHEMBL13158544 0.71
Bromide SCHEMBL7898147 0.71 MEN1 (0.50) ALDH1A1MEN1KMT2AKDM4ELMNA
SCHEMBL10430237 0.71 SLC22A12 (0.42) ALDH1A1MEN1KMT2AKCNH2CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109689664-A The quinoline and azepine quinoline compound that tricyclic heteroaryl as PAR4 inhibitor replaces 百时美施贵宝公司 2019-04-26 CN disclosed