SCHEMBL28286745

SCHEMBL28286745

COC(=O)[C@@H](CCC(=O)C1CCCCC1)NC(=O)OC(C)(C)C

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 9/20 0.47
ITGA2B P08514 9/20 0.47
HDAC4 P56524 1/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
CTSK P43235 3/20 0.46
CTSS P25774 2/20 0.46
CACNA1B Q00975 5/20 0.44
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
HTT P42858 1/20 0.41
NFKB1 P19838 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28286746 1.00 ITGB3 (0.47) ITGB3ITGA2BHDAC4HDAC1HDAC6
SCHEMBL22451614 0.91 CYP1A2 (0.52) ITGB3ITGA2BHDAC4HDAC1HDAC6
SCHEMBL20835667 0.88 CTSK (0.49) ITGB3ITGA2BHDAC4HDAC1HDAC6
SCHEMBL20835669 0.88 CTSK (0.49) ITGB3ITGA2BHDAC4HDAC1HDAC6
SCHEMBL30977182 0.86 CYP1A2 (0.54) HDAC4HDAC1HDAC6CTSKCTSS
SCHEMBL30977183 0.86 CYP1A2 (0.54) HDAC4HDAC1HDAC6CTSKCTSS
SCHEMBL22040793 0.83 HDAC4 (0.44) ITGB3ITGA2BHDAC4HDAC1HDAC6
SCHEMBL22039566 0.83 HDAC4 (0.44) ITGB3ITGA2BHDAC4HDAC1HDAC6
SCHEMBL27444793 0.83 CTSK (0.54) ITGB3ITGA2BHDAC4HDAC1HDAC6
SCHEMBL30044916 0.82 CACNA1B (0.55) ITGB3ITGA2BHDAC4HDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109476639-A Pyrrolidin derivatives 橘生药品工业股份有限公司 2019-03-15 CN disclosed