SCHEMBL28290128

SCHEMBL28290128

COC(=O)c1scc([N+](=O)[O-])c1Cl

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.48
COMT P21964 1/20 0.48
SLC10A6 Q3KNW5 1/20 0.42
MAPT P10636 3/20 0.40
POLB P06746 3/20 0.40
VCAM1 P19320 1/20 0.38
KMT2A Q03164 3/20 0.38
MEN1 O00255 2/20 0.38
MAPK1 P28482 2/20 0.38
TDP1 Q9NUW8 1/20 0.38
LMNA P02545 2/20 0.38
RAF1 P04049 1/20 0.38
HPGD P15428 1/20 0.38
GFER P55789 1/20 0.38
PAX8 Q06710 1/20 0.38
PARP14 Q460N5 1/20 0.37
KDM4E B2RXH2 1/20 0.37
PDGFRB P09619 1/20 0.37
FGFR1 P11362 1/20 0.37
PDGFRA P16234 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13545969 0.82 ALDH1A1 (0.49) ALDH1A1COMTSLC10A6MAPTPOLB
SCHEMBL27873028 0.80 ESR2 (0.41) ALDH1A1VCAM1TDP1LMNAHPGD
SCHEMBL1007296 0.77 KMT2A (0.50) ALDH1A1SLC10A6MAPTPOLBKMT2A
SCHEMBL13545970 0.77 ALDH1A1 (0.42) ALDH1A1COMTSLC10A6VCAM1KMT2A
SCHEMBL31411579 0.76 PDGFRB (0.48) ALDH1A1COMTSLC10A6MAPTPOLB
SCHEMBL2987502 0.74 MAPT (0.49) ALDH1A1MAPTPOLBKMT2AMEN1
SCHEMBL15537166 0.74 MAPT (0.42) COMTMAPTPOLBKMT2AMEN1
SCHEMBL1848834 0.73 ALDH1A1 (0.60) ALDH1A1SLC10A6MAPTPOLBKMT2A
SCHEMBL23459705 0.72 COMT (0.52) ALDH1A1COMTSLC10A6MAPTPOLB
SCHEMBL28866506 0.72 COMT (0.46) ALDH1A1COMTSLC10A6MAPTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110294746-A A kind of new ASK1 inhibitor and its application 山东轩竹医药科技有限公司 2019-10-01 CN disclosed
CN-109563094-A Acyclic derivatives, their preparation method and the pharmaceutical composition containing them that new (miscellaneous) aryl replaces 法国施维雅药厂 2019-04-02 CN disclosed
CN-105283443-B Hete rocyclic derivatives and application thereof 株式会社C&C新药研究所 2018-08-17 CN disclosed