SCHEMBL28291326

SCHEMBL28291326

CCc1c(C#N)cnc(Cl)c1C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSNK1A1 P48729 1/20 0.37
CLK4 Q9HAZ1 1/20 0.37
ALDH1A1 P00352 4/20 0.37
NPSR1 Q6W5P4 4/20 0.37
TDP1 Q9NUW8 1/20 0.37
KDM5A P29375 4/20 0.36
KDM4C Q9H3R0 1/20 0.36
MAPK1 P28482 1/20 0.34
KDM4E B2RXH2 3/20 0.34
LMNA P02545 2/20 0.34
HSD17B10 Q99714 1/20 0.34
NPC1 O15118 1/20 0.33
MAPT P10636 1/20 0.33
RAB9A P51151 1/20 0.33
MDM2 Q00987 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
HTT P42858 2/20 0.33
IDH1 O75874 1/20 0.32
AR P10275 2/20 0.32
PGK1 P00558 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28289895 0.82 HTT (0.38) CSNK1A1CLK4ALDH1A1NPSR1TDP1
SCHEMBL20302398 0.77 CSNK1A1 (0.41) CSNK1A1CLK4ALDH1A1NPSR1TDP1
SCHEMBL3067853 0.74 CSNK1A1 (0.36) CSNK1A1CLK4ALDH1A1KDM5AKDM4C
SCHEMBL3826388 0.73 CSNK1A1 (0.41) CSNK1A1CLK4ALDH1A1NPSR1TDP1
SCHEMBL23532534 0.71 GLA (0.38) ALDH1A1NPSR1KDM5AMAPK1KDM4E
SCHEMBL21736899 0.70 PGK1 (0.37) CSNK1A1CLK4ALDH1A1KDM5AKDM4C
SCHEMBL5200520 0.70 USP7 (0.43) CSNK1A1CLK4ALDH1A1KDM5AKDM4C
SCHEMBL21736855 0.70 KDM5A (0.39) ALDH1A1KDM5AKDM4CMAPK1KDM4E
SCHEMBL14554095 0.69 ALDH1A1 (0.49) CSNK1A1CLK4ALDH1A1NPSR1TDP1
SCHEMBL16884625 0.69 LRRK2 (0.37) ALDH1A1NPSR1TDP1KDM5AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109563043-A SUBSTITUTED PYRIDINES AS INHIBITORS OF DNMT1 葛兰素史密斯克莱知识产权发展有限公司 2019-04-02 CN disclosed