SCHEMBL28291585

SCHEMBL28291585

COc1cc(OC)c2c(C(C)OC=O)c[nH]c2c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.37
KDM4E B2RXH2 2/20 0.37
MAPT P10636 1/20 0.37
ABCG2 Q9UNQ0 1/20 0.36
PDE3B Q13370 2/20 0.34
PDE3A Q14432 2/20 0.34
HTR2A P28223 2/20 0.34
HTR2C P28335 2/20 0.34
HTR2B P41595 2/20 0.34
ERN1 O75460 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C19 P33261 1/20 0.34
HTT P42858 1/20 0.33
MTNR1A P48039 2/20 0.32
MTNR1B P49286 2/20 0.32
HTR1A P08908 1/20 0.32
LMNA P02545 1/20 0.31
GAA P10253 1/20 0.31
HPGD P15428 1/20 0.31
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27908800 0.82 MAPT (0.32) KDM4EMAPTLMNAHSD17B10
SCHEMBL27908784 0.81 MTNR1A (0.43) ALDH1A1KDM4EMTNR1AMTNR1BLMNA
SCHEMBL28678155 0.80 HTR2A (0.45) MAPTABCG2HTR2AHTR2CHTR2B
SCHEMBL27908788 0.78 MTNR1A (0.43) ALDH1A1KDM4EMAPTHTR2AHTR2C
SCHEMBL28929780 0.77 ALDH1A1 (0.57) ALDH1A1KDM4EMAPTHTR2AHTR2C
SCHEMBL28672698 0.74 HTR2A (0.59) ALDH1A1KDM4EMAPTHTR2AHTR2C
SCHEMBL9068972 0.74 HTT (0.41) ALDH1A1KDM4EMAPTERN1CYP1A2
SCHEMBL27551542 0.73 KDM4E (0.33) KDM4EMAPTHSD17B10
SCHEMBL24825685 0.73 ALDH1A1 (0.42) ALDH1A1KDM4EMAPTABCG2PDE3B
SCHEMBL27309524 0.72 GPR17 (0.39) CYP1A2CYP2C19MTNR1AMTNR1BGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102952062-A Substituted benzoheterocyclic compounds and preparation method and application thereof INST MEDICINAL BIOTECHNOLOGY 2013-03-06 CN claimed
CN-109748840-A A kind of synthetic method of 2- substituted indole derivative 中国医学科学院药物研究所 2019-05-14 CN disclosed
CN-102952062-B Replace benzo-heterocycle compound and its preparation method and application 中国医学科学院医药生物技术研究所 2016-06-08 CN disclosed
CN-102952062-A Substituted benzoheterocyclic compounds and preparation method and application thereof INST MEDICINAL BIOTECHNOLOGY 2013-03-06 CN disclosed