SCHEMBL28291677

SCHEMBL28291677

O=CC1CNc2ncccc2C1

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 3/20 0.33
GSK3B P49841 1/20 0.31
ALDH1A1 P00352 1/20 0.31
ADRA1A P35348 1/20 0.30
HTR2A P28223 1/20 0.30
HTR2C P28335 1/20 0.30
HTR2B P41595 1/20 0.30
DRD2 P14416 1/20 0.30
DRD3 P35462 1/20 0.30
TRIM24 O15164 1/20 0.30
TRIM33 Q9UPN9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27458227 0.75 GSK3B (0.35) IDH1GSK3BADRA1ATRIM24TRIM33
SCHEMBL16595227 0.74 DRD2 (0.41) IDH1ALDH1A1DRD2DRD3TRIM24
SCHEMBL24096699 0.74 PLAU (0.37) IDH1GSK3BADRA1AHTR2AHTR2C
SCHEMBL20153297 0.74 GSK3B (0.37) IDH1GSK3BALDH1A1ADRA1AHTR2A
SCHEMBL2298946 0.74 MTNR1A (0.44)
Hydrochloric Acid SCHEMBL31277891 0.72 PLAU (0.36) IDH1ADRA1AHTR2AHTR2CHTR2B
SCHEMBL30585791 0.72 IDH1 (0.43) IDH1
SCHEMBL6013246 0.72 IDH1 (0.43) IDH1
SCHEMBL4597831 0.71 DRD2 (0.52) IDH1DRD2DRD3
SCHEMBL28149742 0.71 IDH1 (0.42) IDH1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109745321-A Pharmaceutical composition comprising FGFR4 inhibitor 上海翰森生物医药科技有限公司 2019-05-14 CN disclosed