SCHEMBL28292634

SCHEMBL28292634

NC(=O)Oc1ccnc(C(N)=O)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
OPRK1 P41145 1/20 0.43
KCNH2 Q12809 1/20 0.43
ADORA3 P0DMS8 1/20 0.41
TSHR P16473 1/20 0.41
MC4R P32245 1/20 0.41
ADRA1A P35348 1/20 0.41
MC3R P41968 1/20 0.41
RAF1 P04049 4/20 0.41
CYP4F2 P78329 2/20 0.39
CYP4A11 Q02928 2/20 0.39
MKNK1 Q9BUB5 1/20 0.38
MKNK2 Q9HBH9 1/20 0.38
OPRM1 P35372 2/20 0.37
HTR1A P08908 1/20 0.37
DRD2 P14416 1/20 0.37
HTR2A P28223 1/20 0.37
BRAF P15056 2/20 0.37
KDM4E B2RXH2 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7720510 0.87 OPRK1 (0.45) MEN1KMT2AOPRK1KCNH2ADORA3
SCHEMBL29262259 0.86 MEN1 (0.48) MEN1KMT2AOPRK1KCNH2RAF1
SCHEMBL28294351 0.82 MEN1 (0.44) MEN1KMT2ARAF1BRAFKDM4E
SCHEMBL28292592 0.82 KDR (0.53) MEN1KMT2ARAF1MKNK2BRAF
SCHEMBL28690607 0.82 MEN1 (0.44) MEN1KMT2AOPRK1KCNH2KDM4E
SCHEMBL2624147 0.81 KDM4E (0.54) OPRK1KCNH2KDM4E
SCHEMBL23488363 0.80 PARP10 (0.55) MEN1KMT2AOPRK1KCNH2KDM4E
SCHEMBL4348844 0.80 OPRK1 (0.41) OPRK1KCNH2ADORA3TSHRMC4R
SCHEMBL9572453 0.79 MEN1 (0.53) MEN1KMT2AMKNK1MKNK2KDM4E
SCHEMBL28723866 0.79 KMT2A (0.53) MEN1KMT2AMKNK1MKNK2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN claimed
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN disclosed
CN-109689647-A The compound that bicyclic heteroaryl replaces 百时美施贵宝公司 2019-04-26 CN disclosed