SCHEMBL28292655

SCHEMBL28292655

COc1cnc2[c]cc(Cl)cc2c1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.34
KDM4E B2RXH2 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
CYP11B1 P15538 4/20 0.33
CYP11B2 P19099 4/20 0.33
CYP17A1 P05093 3/20 0.33
EGFR P00533 1/20 0.33
NFE2L2 Q16236 3/20 0.33
NPC1 O15118 4/20 0.33
RAB9A P51151 3/20 0.33
CYP3A4 P08684 2/20 0.33
F2 P00734 1/20 0.33
GLA P06280 1/20 0.33
HPGD P15428 1/20 0.33
CASP3 P42574 1/20 0.33
SENP7 Q9BQF6 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
AHR P35869 1/20 0.32
PDE3B Q13370 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4397001 0.79 NOS1 (0.32) SMN1; SMN2CYP2C9
SCHEMBL4409372 0.73
SCHEMBL4397674 0.73 PLAU (0.33) SMN1; SMN2
SCHEMBL10321126 0.72 CYP1A2 (0.41) ALDH1A1CYP11B1CYP11B2CYP17A1EGFR
SCHEMBL4411598 0.71 CCR1 (0.31)
SCHEMBL4405857 0.68 HTT (0.31)
SCHEMBL4399733 0.68 PLAU (0.32)
SCHEMBL19776056 0.68 ALDH1A1 (0.35) ALDH1A1SMN1; SMN2EGFRNPC1RAB9A
SCHEMBL17913437 0.67 PDGFRB (0.50) ALDH1A1KDM4EEGFRF2GLA
SCHEMBL27759682 0.66 CHRNB2 (0.43) ALDH1A1KDM4ESMN1; SMN2RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109689647-A The compound that bicyclic heteroaryl replaces 百时美施贵宝公司 2019-04-26 CN disclosed