SCHEMBL28292737

SCHEMBL28292737

O=C(CF)c1cc(Cl)ccc1F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.44
MAPK1 P28482 2/20 0.44
HIF1A Q16665 1/20 0.44
TP53 P04637 2/20 0.44
ERCC5 P28715 2/20 0.43
FEN1 P39748 2/20 0.43
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
MRGPRX4 Q96LA9 1/20 0.41
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
KCNMA1 Q12791 1/20 0.41
SMN1; SMN2 Q16637 3/20 0.40
MAPT P10636 3/20 0.40
MEN1 O00255 2/20 0.40
LMNA P02545 2/20 0.40
HPGD P15428 2/20 0.40
HTT P42858 2/20 0.40
RAB9A P51151 2/20 0.40
KMT2A Q03164 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31678827 0.82 GSK3B (0.52) ALDH1A1MAPK1HIF1ATP53ERCC5
SCHEMBL3930687 0.82 GSK3B (0.52) ALDH1A1MAPK1HIF1ATP53ERCC5
SCHEMBL9941981 0.82 KCNH2 (0.50) ALDH1A1MAPK1HIF1ATP53ERCC5
SCHEMBL27764538 0.82 CES2 (0.63) ALDH1A1MAPK1CES2CES1MAPT
SCHEMBL2609241 0.81 NOS2 (0.55) ALDH1A1MAPK1HIF1ATP53ERCC5
SCHEMBL15771617 0.81 ALDH1A1 (0.46) ALDH1A1MAPK1HIF1ATP53ERCC5
SCHEMBL22170840 0.81 ALDH1A1 (0.44) ALDH1A1MAPK1HIF1ATP53ERCC5
SCHEMBL10361689 0.80 ALDH1A1 (0.69) ALDH1A1MAPK1HIF1AERCC5FEN1
SCHEMBL28072667 0.79 ALDH1A1 (0.50) ALDH1A1MAPK1HIF1ATP53CA1
SCHEMBL9692043 0.79 ALDH1A1 (0.50) ALDH1A1MAPK1HIF1ATP53CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109721539-B Pyrazole amide derivative and preparation method and application thereof 天津药物研究院有限公司 2021-07-09 CN disclosed
CN-109721539-A Pyrazole amide analog derivative and its preparation method and application 天津药物研究院有限公司 2019-05-07 CN disclosed