SCHEMBL28292975

SCHEMBL28292975

O=C(O)c1ccc2cncc-2[nH]1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.53
USP2 O75604 1/20 0.53
HPGD P15428 1/20 0.53
HSD17B10 Q99714 1/20 0.53
PIN1 Q13526 1/20 0.41
MKNK1 Q9BUB5 3/20 0.38
MKNK2 Q9HBH9 3/20 0.38
PTPN1 P18031 2/20 0.38
HCAR2 Q8TDS4 1/20 0.35
ALPL P05186 5/20 0.35
CA12 O43570 3/20 0.35
NAPRT Q6XQN6 1/20 0.34
RPA1 P27694 1/20 0.34
ALOX15 P16050 1/20 0.33
NFKB1 P19838 1/20 0.33
BLM P54132 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
TP53 P04637 1/20 0.33
MAPK14 Q16539 1/20 0.33
XDH P47989 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27645695 0.79 MKNK1 (0.51) KDM4EUSP2HPGDHSD17B10PIN1
Hydrochloric Acid SCHEMBL6336712 0.78 MKNK1 (0.50) KDM4EUSP2HPGDHSD17B10PIN1
SCHEMBL23390037 0.74 KDM4E (0.54) KDM4EUSP2HPGDHSD17B10PIN1
SCHEMBL9750144 0.74 KDM4E (0.63) KDM4EUSP2HPGDHSD17B10PIN1
SCHEMBL27666763 0.73 KDM4E (0.62) KDM4EUSP2HPGDHSD17B10PTPN1
SCHEMBL29621704 0.73 KDM4E (0.53) KDM4EUSP2HPGDHSD17B10PIN1
SCHEMBL8341738 0.72 KDM4E (0.67) KDM4EUSP2HPGDHSD17B10PIN1
Hydrochloric Acid SCHEMBL6343159 0.72 KDM4E (0.61) KDM4EUSP2HPGDHSD17B10PTPN1
SCHEMBL70048 0.71 NFKB1 (0.57) KDM4EUSP2HPGDHSD17B10PIN1
SCHEMBL23416987 0.71 KDM4E (0.50) KDM4EUSP2HPGDHSD17B10SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107235975-B The synthetic method of tert-butyl 6- benzyl -4- oxygen subunit octahydro -1H- pyrrolo- [3,4-b] picolinic acid ester 天津药明康德新药开发有限公司 2019-04-30 CN disclosed