Quinoline

Quinoline

SCHEMBL28293017

NC(=O)C1=NCCO1.c1ccc2ncccc2c1

nearest known ligand 0.47

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.47
PARP1 P09874 1/20 0.38
HDAC1 Q13547 2/20 0.38
HDAC2 Q92769 2/20 0.38
HDAC3 O15379 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC7 Q8WUI4 1/20 0.38
HDAC10 Q969S8 1/20 0.38
HDAC11 Q96DB2 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
HDAC9 Q9UKV0 1/20 0.38
HDAC5 Q9UQL6 1/20 0.38
AR P10275 1/20 0.37
NPC1 O15118 2/20 0.36
POLB P06746 2/20 0.36
RAB9A P51151 1/20 0.36
KDM4E B2RXH2 2/20 0.35
MEN1 O00255 2/20 0.35
MAPT P10636 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Quinoline SCHEMBL28292999 0.87 ALDH1A1 (0.49) ALDH1A1HDAC1HDAC2HDAC3HDAC4
Quinoline SCHEMBL28140139 0.78 ALDH1A1 (0.55) ALDH1A1NPC1POLBRAB9AKDM4E
Quinoline SCHEMBL28144363 0.78 ALDH1A1 (0.55) ALDH1A1HDAC8NPC1POLBRAB9A
Quinoline SCHEMBL28213101 0.77 ALDH1A1 (0.53) ALDH1A1NPC1POLBRAB9AKDM4E
Quinoline SCHEMBL5272119 0.77 ALDH1A1 (0.74) ALDH1A1PARP1HDAC1HDAC2NPC1
Quinoline SCHEMBL1287895 0.77 ALDH1A1 (0.74) ALDH1A1PARP1HDAC1HDAC2NPC1
Quinoline SCHEMBL2201840 0.77 ALDH1A1 (0.74) ALDH1A1PARP1HDAC1HDAC2NPC1
Quinoline SCHEMBL27782946 0.75 ALDH1A1 (0.71) ALDH1A1PARP1HDAC1HDAC2NPC1
Quinoline SCHEMBL28318728 0.75 ALDH1A1 (0.55) ALDH1A1NPC1POLBRAB9AKDM4E
Quinoline SCHEMBL28087657 0.74 ALDH1A1 (0.50) ALDH1A1NPC1POLBRAB9AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109641886-A bicyclic BET bromodomain inhibitors and uses thereof 康威基内有限公司 2019-04-16 CN claimed
CN-109641886-A bicyclic BET bromodomain inhibitors and uses thereof 康威基内有限公司 2019-04-16 CN disclosed