Quinoline

Quinoline

SCHEMBL28292999

O=C(O)C1=NCCO1.c1ccc2ncccc2c1

nearest known ligand 0.49

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.49
MCL1 Q07820 1/20 0.41
HDAC3 O15379 1/20 0.41
HDAC4 P56524 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC7 Q8WUI4 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC10 Q969S8 1/20 0.41
HDAC11 Q96DB2 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
HDAC9 Q9UKV0 1/20 0.41
HDAC5 Q9UQL6 1/20 0.41
MGAM O43451 2/20 0.39
PABPC1 P11940 1/20 0.38
NPC1 O15118 3/20 0.37
POLB P06746 2/20 0.37
RAB9A P51151 1/20 0.37
CYP3A4 P08684 1/20 0.36
MEN1 O00255 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Quinoline SCHEMBL28293017 0.87 ALDH1A1 (0.47) ALDH1A1MCL1HDAC3HDAC4HDAC1
Benzene SCHEMBL28149443 0.79 HDAC3 (0.43) ALDH1A1HDAC3HDAC4HDAC1HDAC7
Quinoline SCHEMBL28144363 0.79 ALDH1A1 (0.55) ALDH1A1MCL1HDAC8PABPC1NPC1
Quinoline SCHEMBL28318728 0.76 ALDH1A1 (0.55) ALDH1A1NPC1POLBRAB9ACYP3A4
Quinoline SCHEMBL28140139 0.76 ALDH1A1 (0.55) ALDH1A1NPC1POLBRAB9ACYP3A4
Quinoline SCHEMBL372690 0.76 ALDH1A1 (0.77) ALDH1A1MCL1MGAMPABPC1NPC1
Quinoline SCHEMBL5874493 0.76 ALDH1A1 (0.77) ALDH1A1MCL1MGAMPABPC1NPC1
Quinoline SCHEMBL5283313 0.76 ALDH1A1 (0.77) ALDH1A1MCL1MGAMPABPC1NPC1
SCHEMBL1030035 0.76
Quinoline SCHEMBL28213101 0.75 ALDH1A1 (0.53) ALDH1A1NPC1POLBRAB9ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109641886-A bicyclic BET bromodomain inhibitors and uses thereof 康威基内有限公司 2019-04-16 CN disclosed