SCHEMBL28293549

SCHEMBL28293549

CN1CCN(c2ccc([N+](=O)[O-])cc2C(=O)c2ccccc2)CC1.Nc1cncnc1N

nearest known ligand 0.73

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 14/20 0.73
LMNA P02545 10/20 0.73
GAA P10253 2/20 0.73
KMT2A Q03164 2/20 0.60
CYP1A2 P05177 2/20 0.60
CYP3A4 P08684 2/20 0.60
CYP2C9 P11712 2/20 0.60
CYP2C19 P33261 2/20 0.60
MEN1 O00255 1/20 0.60
CYP2D6 P10635 1/20 0.60
SMN1; SMN2 Q16637 4/20 0.59
MAPT P10636 4/20 0.59
HTT P42858 3/20 0.59
POLB P06746 2/20 0.59
KDM4E B2RXH2 1/20 0.58
WDR5 P61964 1/20 0.52
PAX8 Q06710 3/20 0.49
RAB9A P51151 1/20 0.48
MAPK1 P28482 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28293598 0.89 ALDH1A1 (0.73) ALDH1A1LMNAGAAKMT2ACYP1A2
SCHEMBL28291864 0.87 ALDH1A1 (0.76) ALDH1A1LMNAGAAKMT2ACYP1A2
SCHEMBL28872862 0.86 ALDH1A1 (0.80) ALDH1A1LMNAGAAKMT2ACYP1A2
SCHEMBL27954071 0.86 ALDH1A1 (1.00) ALDH1A1LMNAGAAKMT2ACYP1A2
Methyl Alcohol SCHEMBL28334259 0.84 ALDH1A1 (0.98) ALDH1A1LMNAGAAKMT2ACYP1A2
Acetic Acid SCHEMBL27840869 0.84 ALDH1A1 (0.95) ALDH1A1LMNAGAAKMT2ACYP1A2
Diaminopyrimidine SCHEMBL28291871 0.81 ALDH1A1 (0.74) ALDH1A1LMNAGAAKMT2ACYP1A2
SCHEMBL1972566 0.73 ALDH1A1 (0.75) ALDH1A1LMNAGAAKMT2ACYP1A2
SCHEMBL10732007 0.73 ALDH1A1 (0.77) ALDH1A1LMNAGAAKMT2ACYP1A2
SCHEMBL8440614 0.73 LMNA (0.80) ALDH1A1LMNAGAAKMT2ACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109734674-A Phenyl amines WDR5 protein-protein interaction inhibitor and its preparation method and purposes 中国药科大学 2019-05-10 CN disclosed