SCHEMBL28293920

SCHEMBL28293920

COC(=O)CC(NC(=O)OC(C)(C)C)c1ccccc1Br

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSS P25774 4/20 0.45
CTSK P43235 3/20 0.45
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
HTT P42858 3/20 0.42
RAB9A P51151 2/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
NPC1 O15118 1/20 0.42
MAPT P10636 2/20 0.42
ALDH1A1 P00352 1/20 0.42
LMNA P02545 1/20 0.42
TP53 P04637 1/20 0.42
PKM P14618 1/20 0.42
HPGD P15428 1/20 0.42
TSHR P16473 1/20 0.42
AGTR1 P30556 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
HSD17B10 Q99714 1/20 0.42
CYP26A1 O43174 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28265926 1.00 CTSS (0.45) CTSSCTSKCYP2C9CYP2C19HTT
SCHEMBL27886474 1.00 CTSS (0.45) CTSSCTSKCYP2C9CYP2C19HTT
SCHEMBL19744342 0.88 CYP26A1 (0.53) CTSSCTSKHTTRAB9AMEN1
SCHEMBL19744343 0.88 CYP26A1 (0.53) CTSSCTSKHTTRAB9AMEN1
SCHEMBL3447780 0.86 CACNA1B (0.47) CTSSCTSKHTTRAB9AMAPT
SCHEMBL24198500 0.85 CTSS (0.47) CTSSCTSKHTTRAB9AMEN1
SCHEMBL5768896 0.85 RAB9A (0.45) HTTRAB9AMEN1KMT2AMAPT
SCHEMBL3447675 0.85 CTSS (0.45) CTSSCTSKHTTRAB9AMEN1
SCHEMBL5862217 0.81 CTSK (0.52) CTSSCTSKHTTRAB9AMEN1
SCHEMBL31633773 0.81 CTSK (0.52) CTSSCTSKHTTRAB9AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109678859-B Dihydropyrimidine compound and application thereof in medicine 广东东阳光药业有限公司 2020-12-29 CN disclosed
CN-109678859-A Dihydropyrimidines and its application in drug 广东东阳光药业有限公司 2019-04-26 CN disclosed