SCHEMBL28294290

SCHEMBL28294290

NC(=O)Oc1ccc(C(=O)N2CCOC[C@@H]2CO)nc1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 2/20 0.40
FPR2 P25090 1/20 0.40
LRRK2 Q5S007 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
TRPC6 Q9Y210 5/20 0.39
SMN1; SMN2 Q16637 1/20 0.38
PDK1 Q15118 1/20 0.37
ROCK2 O75116 1/20 0.36
ROCK1 Q13464 1/20 0.36
NTRK1 P04629 2/20 0.36
MTOR P42345 3/20 0.35
HCRTR1 O43613 3/20 0.35
HCRTR2 O43614 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28941116 1.00 SCN9A (0.40) SCN9AFPR2LRRK2MEN1KMT2A
SCHEMBL28941054 1.00 SCN9A (0.40) SCN9AFPR2LRRK2MEN1KMT2A
SCHEMBL28872982 0.78 SMN1; SMN2 (0.62) SCN9ASMN1; SMN2MTOR
SCHEMBL28941055 0.77 NTRK1 (0.41) LRRK2MEN1KMT2ASMN1; SMN2PDK1
SCHEMBL28294291 0.77 NTRK1 (0.41) LRRK2MEN1KMT2ASMN1; SMN2PDK1
SCHEMBL28941108 0.77 NTRK1 (0.41) LRRK2MEN1KMT2ASMN1; SMN2PDK1
SCHEMBL28292565 0.76 L3MBTL1 (0.49) SMN1; SMN2PDK1NTRK1HCRTR1HCRTR2
SCHEMBL28941103 0.75 SCN9A (0.49) SCN9ALRRK2KMT2ASMN1; SMN2PDK1
SCHEMBL28941076 0.75 SCN9A (0.49) SCN9ALRRK2KMT2ASMN1; SMN2PDK1
SCHEMBL28940980 0.72 SCN9A (0.48) SCN9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN claimed
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN disclosed
CN-109689647-A The compound that bicyclic heteroaryl replaces 百时美施贵宝公司 2019-04-26 CN disclosed