SCHEMBL28940980

SCHEMBL28940980

NC(=O)Oc1ccc(C(=O)N2CC[C@@H](CO)C2)nc1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 3/20 0.48
GRM3 Q14832 3/20 0.43
VNN1 O95497 1/20 0.42
LIPE Q05469 1/20 0.40
DRD3 P35462 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.39
L3MBTL3 Q96JM7 1/20 0.39
HRH3 Q9Y5N1 3/20 0.39
KCNH2 Q12809 1/20 0.39
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
KMT2A Q03164 1/20 0.38
KDM5A P29375 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28294359 1.00 SCN9A (0.48) SCN9AGRM3VNN1LIPEDRD3
SCHEMBL28292616 0.84 SCN9A (0.46) SCN9AGRM3VNN1DRD3L3MBTL1
SCHEMBL28292584 0.84 SCN9A (0.46) SCN9AGRM3VNN1DRD3L3MBTL1
SCHEMBL28941103 0.82 SCN9A (0.49) SCN9ADRD3HRH3KCNH2KMT2A
SCHEMBL28941076 0.82 SCN9A (0.49) SCN9ADRD3HRH3KCNH2KMT2A
SCHEMBL28294319 0.82 HRH3 (0.47) SCN9AGRM3LIPEDRD3L3MBTL1
SCHEMBL28292599 0.80 KMT2A (0.52) SCN9AGRM3VNN1L3MBTL1L3MBTL3
SCHEMBL28292628 0.80 KMT2A (0.52) SCN9AGRM3VNN1L3MBTL1L3MBTL3
SCHEMBL28940974 0.80 KMT2A (0.52) SCN9AGRM3VNN1L3MBTL1L3MBTL3
SCHEMBL21379649 0.75 VNN1 (0.45) SCN9AVNN1L3MBTL1L3MBTL3NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN claimed
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN disclosed