SCHEMBL28294319

SCHEMBL28294319

NC(=O)Oc1ccc(C(=O)N2CCC(O)CC2)nc1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 7/20 0.47
KCNH2 Q12809 1/20 0.47
L3MBTL3 Q96JM7 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
GRM3 Q14832 1/20 0.44
SCN9A Q15858 2/20 0.44
DRD3 P35462 1/20 0.44
TRPC6 Q9Y210 2/20 0.43
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.41
LIPE Q05469 1/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
MAPK7 Q13164 1/20 0.40
HPGD P15428 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28292584 0.92 SCN9A (0.46) HRH3KCNH2L3MBTL3L3MBTL1GRM3
SCHEMBL28292616 0.92 SCN9A (0.46) HRH3KCNH2L3MBTL3L3MBTL1GRM3
SCHEMBL28292599 0.85 KMT2A (0.52) HRH3KCNH2L3MBTL3L3MBTL1GRM3
SCHEMBL28940974 0.85 KMT2A (0.52) HRH3KCNH2L3MBTL3L3MBTL1GRM3
SCHEMBL28292628 0.85 KMT2A (0.52) HRH3KCNH2L3MBTL3L3MBTL1GRM3
SCHEMBL28872982 0.83 SMN1; SMN2 (0.62) HRH3SCN9ADRD3NPC1RAB9A
SCHEMBL28940980 0.82 SCN9A (0.48) HRH3KCNH2L3MBTL3L3MBTL1GRM3
SCHEMBL28294359 0.82 SCN9A (0.48) HRH3KCNH2L3MBTL3L3MBTL1GRM3
SCHEMBL31262623 0.76 L3MBTL1 (0.50) HRH3KCNH2L3MBTL3L3MBTL1SCN9A
SCHEMBL20254511 0.76 L3MBTL1 (0.50) HRH3KCNH2L3MBTL3L3MBTL1SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN claimed
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN disclosed
CN-109689647-A The compound that bicyclic heteroaryl replaces 百时美施贵宝公司 2019-04-26 CN disclosed