SCHEMBL2829443

SCHEMBL2829443

O=C(Nc1cccc(Cl)c1)Oc1ncsc1NC1CCCC1

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.50
KMT2A Q03164 3/20 0.50
EPHX2 P34913 3/20 0.50
LMNA P02545 2/20 0.50
NPC1 O15118 2/20 0.50
RAB9A P51151 2/20 0.50
EPHX1 P07099 2/20 0.50
TSHR P16473 1/20 0.50
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C19 P33261 1/20 0.45
HTT P42858 1/20 0.44
MAPT P10636 2/20 0.43
HPGD P15428 1/20 0.42
ALOX15 P16050 1/20 0.42
GRM5 P41594 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2832981 0.99 EPHX2 (0.52) MEN1KMT2AEPHX2LMNANPC1
SCHEMBL2826660 0.96 LMNA (0.46) MEN1KMT2AEPHX2LMNANPC1
SCHEMBL2831135 0.88 NPC1 (0.51) KMT2ANPC1RAB9ACYP3A4MAPT
SCHEMBL2828482 0.87 NPC1 (0.50) MEN1KMT2ANPC1RAB9AMAPT
SCHEMBL2828420 0.87 GRK2 (0.44) MEN1KMT2ANPC1RAB9AHTT
SCHEMBL2830068 0.87 SMN1; SMN2 (0.44) MEN1KMT2AEPHX2LMNARAB9A
SCHEMBL2826937 0.84 ALDH1A1 (0.48) KMT2ANPC1RAB9ACYP3A4HPGD
SCHEMBL2830058 0.83 LMNA (0.50) MEN1KMT2ALMNANPC1RAB9A
SCHEMBL2829765 0.83 KMT2A (0.43) MEN1KMT2ALMNANPC1RAB9A
SCHEMBL2825247 0.83 NPC1 (0.44) MEN1KMT2ALMNANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1844044-B1 THIAZOLE-4-CARBOXAMIDE DERIVATIVES AS MGLUR5 ANTAGONISTS HOFFMANN LA ROCHE (CH) 2010-07-21 EP claimed